SCHEMBL17848588

SCHEMBL17848588

FCOc1cccc(OCCBr)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
MAPK1 P28482 2/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
PRSS1 P07477 6/20 0.37
KCNA3 P22001 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
TSHR P16473 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
HIF1A Q16665 1/20 0.36
CHRNB2 P17787 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8155382 0.89 SMN1; SMN2 (0.50) SMN1; SMN2NPC1MAPTRAB9AMAPK1
SCHEMBL4737237 0.85 TP53 (0.45) SMN1; SMN2MAPK1MTNR1AMTNR1BMAOB
SCHEMBL19439532 0.80 MAPT (0.66) SMN1; SMN2NPC1MAPTRAB9AMAPK1
SCHEMBL1770655 0.80 MAPK1 (0.61) MAPK1MTNR1AMTNR1BMAOBCYP1A2
SCHEMBL5726997 0.80 MAPK1 (0.56) MAPTRAB9AMAPK1CYP1A2CYP2D6
SCHEMBL1497882 0.80 MAOB (0.49) SMN1; SMN2NPC1MAPTRAB9AMAOA
SCHEMBL30674601 0.80 MAPK1 (0.61) MAPK1MTNR1AMTNR1BMAOBCYP1A2
SCHEMBL30044154 0.80 MAOB (0.49) SMN1; SMN2NPC1MAPTRAB9AMAOA
SCHEMBL7614389 0.80 KMT2A (0.54) SMN1; SMN2NPC1MAPTRAB9AMAPK1
SCHEMBL3720181 0.79 CETP (0.42) SMN1; SMN2NPC1MAPTRAB9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
WO-2016100940-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2016-06-23 WO disclosed