SCHEMBL17848804

SCHEMBL17848804

CC(C)C(=O)C(C)C.CCOc1cc([C@@H](CS(C)(=O)=O)N2C(=O)c3cccc(CC(N)=O)c3C2=O)ccc1OC

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 20/20 0.75
PDE4C Q08493 19/20 0.75
PDE4A P27815 13/20 0.75
PDE4D Q08499 13/20 0.75
HTR2B P41595 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17848801 0.97 PDE4B (0.79) PDE4BPDE4CPDE4APDE4DHTR2B
SCHEMBL22029271 0.97 PDE4B (0.79) PDE4BPDE4CPDE4APDE4DHTR2B
Acetone SCHEMBL17848799 0.96 PDE4B (0.76) PDE4BPDE4CPDE4APDE4DHTR2B
Alcohol SCHEMBL17848800 0.96 PDE4B (0.77) PDE4BPDE4CPDE4APDE4DHTR2B
Isobutyraldehyde SCHEMBL17848805 0.94 PDE4B (0.72) PDE4BPDE4CPDE4APDE4DHTR2B
Propanol SCHEMBL17848792 0.94 PDE4B (0.74) PDE4BPDE4CPDE4APDE4DHTR2B
SCHEMBL30626414 0.91 PDE4B (0.77) PDE4BPDE4CPDE4APDE4DHTR2B
SCHEMBL28672780 0.91 PDE4B (0.77) PDE4BPDE4CPDE4APDE4DHTR2B
SCHEMBL7401395 0.89 PDE4B (0.76) PDE4BPDE4CPDE4APDE4DHTR2B
SCHEMBL537193 0.88 PDE4B (0.83) PDE4BPDE4CPDE4APDE4DHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016097156-A1 NOVEL SOLVATES OF N-[2-[(1S)-1-(3-ETHOXY-4-METHOXYPHENYL)-2-(METHYLSULFONYL)ETHYL]-2,3-DIHYDRO-1,3-DIOXO-1H-ISOINDOL-4-YL]ACETAMIDE LEK PHARMACEUTICALS D.D. (SI) 2016-06-23 WO disclosed