SCHEMBL17848940

SCHEMBL17848940

C[SiH](O[C@@H]1CC(c2cc(F)ccc2F)N(C(=O)OC(C)(C)C)C1)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 14/20 0.41
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
GPR119 Q8TDV5 1/20 0.35
JAK2 O60674 1/20 0.35
TACR1 P25103 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18588956 0.84 NR1H2 (0.42) NTRK1NR1H2NR1H3GPR119JAK2
SCHEMBL16293086 0.83 NTRK1 (0.41) NTRK1NR1H2NR1H3GPR119JAK2
SCHEMBL15017396 0.83 NTRK1 (0.41) NTRK1NR1H2NR1H3GPR119JAK2
SCHEMBL18878036 0.83 NTRK1 (0.45) NTRK1NR1H2NR1H3GPR119JAK2
SCHEMBL17821020 0.83 CYP1A2 (0.44) NTRK1NR1H2NR1H3GPR119JAK2
SCHEMBL23083856 0.83 NTRK1 (0.44) NTRK1NR1H2NR1H3GPR119
SCHEMBL18588911 0.83 CYP1A2 (0.44) NTRK1NR1H2NR1H3GPR119JAK2
SCHEMBL17820748 0.83 NTRK1 (0.44) NTRK1NR1H2NR1H3GPR119
SCHEMBL17820744 0.83 NTRK1 (0.44) NTRK1NR1H2NR1H3GPR119
SCHEMBL18588910 0.83 CYP1A2 (0.44) NTRK1NR1H2NR1H3GPR119JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233863-A1 FUSED RING HETEROARYL COMPOUNDS AND THEIR USE AS TRK INHIBITORS CMG Pharmaceutical Co., Ltd. (KR) 2017-10-25 EP disclosed
WO-2016097869-A1 FUSED RING HETEROARYL COMPOUNDS AND THEIR USE AS TRK INHIBITORS CMG PHARMACEUTICAL CO., LTD. (KR) 2016-06-23 WO disclosed