SCHEMBL17850211

SCHEMBL17850211

CN1/C(=N\C(=O)OC(C)(C)C)N[C@](C)(c2cc(N)cc(F)c2)CS1(=O)=O

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10328997 1.00 BACE1 (0.31) BACE1BACE2
SCHEMBL10328658 0.85 BACE1 (0.32) BACE1BACE2
SCHEMBL15721339 0.85 BACE1 (0.32) BACE1BACE2
SCHEMBL15895194 0.85
SCHEMBL10328636 0.85
SCHEMBL10328683 0.84 BACE1 (0.34) BACE1BACE2
SCHEMBL15892961 0.84 BACE1 (0.34) BACE1BACE2
SCHEMBL10328681 0.82 BACE1 (0.39) BACE1BACE2
SCHEMBL15895228 0.82 BACE1 (0.34) BACE1BACE2
SCHEMBL10328668 0.82 BACE1 (0.34) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3034080-A1 IMINOTHIADIAZINE DIOXIDE COMPOUNDS AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE Merck Sharp & Dohme Corp. (US) 2016-06-22 EP disclosed