SCHEMBL17850455

SCHEMBL17850455

CCc1ccc(-n2cc(-c3n[nH]c4ccccc34)nn2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
CDC7 O00311 2/20 0.44
ROCK2 O75116 2/20 0.44
MAP4K4 O95819 2/20 0.44
PIM1 P11309 2/20 0.44
CDK2 P24941 2/20 0.44
HIPK2 Q9H2X6 2/20 0.44
IRAK4 Q9NWZ3 2/20 0.44
LRRK2 Q5S007 1/20 0.43
PTGS2 P35354 3/20 0.42
FLT3 P36888 3/20 0.41
S1PR1 P21453 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALPL P05186 1/20 0.41
GAA P10253 1/20 0.41
IDO1 P14902 1/20 0.41
HPGD P15428 1/20 0.41
TTK P33981 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10194704 0.88 GRM4 (0.46) GRM4CDC7ROCK2MAP4K4PIM1
SCHEMBL9951736 0.88 GRM4 (0.46) GRM4CDC7ROCK2MAP4K4PIM1
Hydrochloric Acid SCHEMBL9952647 0.86 GRM4 (0.45) GRM4CDC7ROCK2MAP4K4PIM1
Ammonia Solution, Strong SCHEMBL27926209 0.85 FLT3 (0.56) GRM4ADORA3CDC7ROCK2MAP4K4
Hydrochloric Acid SCHEMBL28806324 0.84 FLT3 (0.54) GRM4ADORA3CDC7ROCK2MAP4K4
SCHEMBL9951780 0.83 GRM4 (0.45) GRM4CDC7ROCK2MAP4K4PIM1
SCHEMBL10195754 0.83 GRM4 (0.49) GRM4CDC7ROCK2MAP4K4PIM1
SCHEMBL9951926 0.83 OGT (0.43) GRM4CDC7ROCK2MAP4K4PIM1
SCHEMBL10196818 0.82 GRM4 (0.46) GRM4CDC7ROCK2MAP4K4PIM1
SCHEMBL9952315 0.82 GRM4 (0.44) GRM4CDC7ROCK2MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655357-B1 INDAZOLYL TRIAZOLE DERIVATIVES AS IRAK INHIBITORS MERCK SERONO SA (CH) 2016-06-22 EP disclosed