SCHEMBL17865818

SCHEMBL17865818

COc1cc([C@@H](CN2CCC2)Nc2ncnc3c(OC(N)=O)cccc23)ccc1F

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 16/20 0.66
AKT1 P31749 13/20 0.66
AURKB Q96GD4 12/20 0.66
INCENP Q9NQS7 10/20 0.66
AURKA O14965 4/20 0.53
AKT2 P31751 1/20 0.51
AKT3 Q9Y243 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17865819 0.92 RPS6KB1 (0.78) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL17865856 0.91 RPS6KB1 (0.60) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL8511555 0.90 RPS6KB1 (0.81) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL8589247 0.90 RPS6KB1 (0.81) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL17865843 0.89 RPS6KB1 (0.62) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL17865845 0.89 AKT1 (0.67) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL17865853 0.89 AKT1 (0.69) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL17865808 0.88 RPS6KB1 (0.61) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL17865864 0.88 AKT1 (0.78) RPS6KB1AKT1AURKBINCENPAURKA
SCHEMBL17865847 0.88 AKT1 (0.79) RPS6KB1AKT1AURKBINCENPAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2643313-B9 QUINAZOLINE CARBOXAMIDE AZETIDINES MERCK PATENT GMBH (DE) 2017-02-22 EP claimed
EP-2643313-B1 QUINAZOLINE CARBOXAMIDE AZETIDINES MERCK PATENT GMBH (DE) 2016-06-29 EP claimed