SCHEMBL17875305

SCHEMBL17875305

Cn1[nH]c2ccc([N+](=O)[O-])cc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.56
CA9 Q16790 2/20 0.56
ALOX5 P09917 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
CTSV O60911 2/20 0.48
CTSL P07711 2/20 0.48
PARP1 P09874 2/20 0.48
GRIA1 P42261 1/20 0.47
GRIA2 P42262 1/20 0.47
GRIA3 P42263 1/20 0.47
GRIA4 P48058 1/20 0.47
MAPT P10636 4/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 2/20 0.46
POLB P06746 1/20 0.46
PKM P14618 1/20 0.46
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16138106 0.87 DAO (0.53) CA12CA9ALOX5L3MBTL1CTSV
SCHEMBL8834687 0.83 KDM4E (0.53) CA12CA9L3MBTL1PARP1GRIA1
SCHEMBL10998454 0.78 CA12 (0.69) CA12CA9L3MBTL1CTSVCTSL
SCHEMBL16007675 0.76 CA12 (0.58) CA12CA9L3MBTL1CTSVCTSL
Tert-Butyl Formate SCHEMBL28043656 0.76 DAO (0.42) CA12CA9ALOX5L3MBTL1CTSV
SCHEMBL31482838 0.74 MAPT (0.53) CA12CA9L3MBTL1PARP1GRIA1
SCHEMBL31482835 0.74 MAPT (0.53) CA12CA9L3MBTL1PARP1GRIA1
SCHEMBL3648969 0.74 MAPT (0.53) CA12CA9L3MBTL1PARP1GRIA1
SCHEMBL7431126 0.72 CA12 (0.64) CA12CA9L3MBTL1CTSVCTSL
SCHEMBL17434518 0.72 CA12 (0.64) CA12CA9L3MBTL1CTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2710013-B1 NOVEL COMPOUNDS AS DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2016-06-29 EP disclosed