SCHEMBL17878207

SCHEMBL17878207

C[C@@H]1CC[C@@H](N)CN1C(=O)c1ccccc1N/N=C\C=N

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HCRTR2 O43614 15/20 0.38
TSHR P16473 1/20 0.36
HCRTR1 O43613 9/20 0.35
PIK3CD O00329 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19652346 0.91 NPSR1 (0.38) NPSR1MEN1KMT2AHCRTR2TSHR
SCHEMBL17863848 0.86 NPSR1 (0.40) NPSR1MEN1KMT2AHCRTR2TSHR
SCHEMBL19604257 0.85 NPSR1 (0.39) NPSR1MEN1KMT2AHCRTR2TSHR
SCHEMBL17724395 0.84 NPSR1 (0.56) NPSR1MEN1KMT2ATSHR
SCHEMBL27055106 0.84 NPSR1 (0.55) NPSR1MEN1KMT2ATSHR
SCHEMBL19574012 0.82 HCRTR2 (0.43) MEN1KMT2AHCRTR2HCRTR1
SCHEMBL17856314 0.81 PARP1 (0.40) MEN1KMT2ATSHR
SCHEMBL19604256 0.78 HCRTR2 (0.48) HCRTR2HCRTR1
SCHEMBL19604254 0.75 HCRTR2 (0.64) HCRTR2HCRTR1
SCHEMBL19604255 0.75 HCRTR2 (0.64) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016106106-A2 FUSED HETEROARYL DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-30 WO disclosed