SCHEMBL17895160

SCHEMBL17895160

CC(C)(C)[Si](OC[C@@H]1CO[C@@H](CO)CN1C(=O)O)(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 3/20 0.38
MGAM O43451 3/20 0.34
CYP3A4 P08684 3/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
NR3C2 P08235 1/20 0.30
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17895054 0.90 SRC (0.38) SMYD2
SCHEMBL31410012 0.90 SRC (0.38) SMYD2
SCHEMBL14636816 0.90 SRC (0.38) SMYD2
SCHEMBL14636814 0.90 SRC (0.38) SMYD2
SCHEMBL17894245 0.82 MGAM (0.38) SMYD2MGAM
SCHEMBL31409894 0.82 MGAM (0.38) SMYD2MGAM
SCHEMBL15877751 0.82 MGAM (0.38) SMYD2MGAM
SCHEMBL15577547 0.82
SCHEMBL15577715 0.81 SMYD2 (0.35) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL18170178 0.80 SMYD2 (0.36) SMYD2MGAMCYP3A4HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3240543-B1 BTK INHIBITORS MERCK SHARP & DOHME LLC (US) 2024-11-06 EP disclosed
WO-2016106628-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-07-07 WO disclosed