SCHEMBL17896789

SCHEMBL17896789

CN1CCCC(Cc2cnccn2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.50
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
CDC42BPB Q9Y5S2 1/20 0.43
CHRM2 P08172 4/20 0.42
CHRM1 P11229 4/20 0.42
CHRM3 P20309 3/20 0.42
KCNH2 Q12809 3/20 0.39
ADRA2A P08913 2/20 0.39
DRD1 P21728 2/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
ADRA1A P35348 2/20 0.39
OPRM1 P35372 2/20 0.39
DRD3 P35462 2/20 0.39
HRH3 Q9Y5N1 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896377 0.83 MAP4K4 (0.47) MAP4K4ROCK2ROCK1CDC42BPBCHRM2
SCHEMBL12090380 0.79 KCNH2 (0.53) MAP4K4CHRM2CHRM1CHRM3KCNH2
SCHEMBL3507744 0.79 HRH4 (0.44) MAP4K4HRH3LMNATSHRHTR6
SCHEMBL25235377 0.76 MAP4K4 (0.40) MAP4K4HRH3LMNAVNN1JAK2
SCHEMBL12090436 0.75 CHRM2 (0.64) CHRM2CHRM1CHRM3HRH3
SCHEMBL12090334 0.74 MAP4K4 (0.47) MAP4K4CHRM2CHRM1CHRM3KCNH2
SCHEMBL27022433 0.74 MAP4K4 (0.38) MAP4K4OPRM1LMNA
SCHEMBL23206055 0.73 HRH3 (0.49) MAP4K4CHRM2CHRM1CHRM3KCNH2
SCHEMBL13452390 0.73 CHRM2 (0.45) ROCK2ROCK1CDC42BPBCHRM2CHRM1
SCHEMBL20893003 0.72 KMT2A (0.50) TSHRVNN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382241-B2 Aminoquinazoline and pyridopyrimidine derivatives GENENTECH, INC. (US) 2016-07-05 US disclosed