SCHEMBL17897906

SCHEMBL17897906

C#CCCCn1c(Sc2ccccc2C)nc2c(N)ncnc21

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90B1 P14625 16/20 0.79
HSP90AA1 P07900 11/20 0.78
HSP90AB1 P08238 11/20 0.78
TRAP1 Q12931 5/20 0.78
ERBB2 P04626 2/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17897912 0.88 HSP90B1 (1.00) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL17897923 0.88 HSP90B1 (1.00) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL17897930 0.88 HSP90B1 (1.00) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL17900410 0.87 HSP90B1 (1.00) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL16486526 0.87 HSP90B1 (0.78) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL21861895 0.86 HSP90B1 (0.80) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL17897917 0.86 HSP90B1 (0.82) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL17897928 0.86 HSP90B1 (1.00) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2
SCHEMBL16512927 0.85 HSP90B1 (0.80) HSP90B1HSP90AA1HSP90AB1TRAP1
SCHEMBL16487078 0.84 HSP90B1 (0.85) HSP90B1HSP90AA1HSP90AB1TRAP1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230123747-A1 SELECTIVE GRP94 INHIBITORS AND USES THEREOF MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2023-04-20 US disclosed
US-20200102312-A1 SELECTIVE GRP94 INHIBITORS AND USES THEREOF MEMORIAL SLOAN-KETTERING CANCER CENTER 2020-04-02 US disclosed
US-10421758-B2 Selective Grp94 inhibitors and uses thereof MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2019-09-24 US disclosed
US-20160194328-A1 SELECTIVE GRP94 INHIBITORS AND USES THEREOF MEMORIAL SLOAN-KETTERING CANCER CENTER 2016-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160194328-A1 SELECTIVE GRP94 INHIBITORS AND USES THEREOF HSP90B1, HSP90AB2P, HSPE1 HSP90B1 1/4885HSP90AA1 9/4885HSP90AB1 4/4885
US-10421758-B2 Selective Grp94 inhibitors and uses thereof HSP90B1, HSP90AB2P, HSPE1 HSP90B1 1/4885HSP90AA1 9/4885HSP90AB1 4/4885
US-20200102312-A1 SELECTIVE GRP94 INHIBITORS AND USES THEREOF HSP90B1, HSP90AB2P, HSPE1 HSP90B1 1/4885HSP90AA1 9/4885HSP90AB1 4/4885
US-20230123747-A1 SELECTIVE GRP94 INHIBITORS AND USES THEREOF HSP90B1, HSP90AB2P, HSPE1 HSP90B1 1/4885HSP90AA1 9/4885HSP90AB1 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.