SCHEMBL17934367

SCHEMBL17934367

COCC(C)Oc1cc2ncnc(Cl)c2c2c1OCCO2

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.63
KDR P35968 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17934406 0.86 EGFR (0.58) EGFRKDR
SCHEMBL17934387 0.85 EGFR (0.59) EGFRKDR
SCHEMBL17934351 0.83 EGFR (0.60) EGFRKDR
SCHEMBL21750829 0.82 EGFR (0.45) EGFRKDR
SCHEMBL21750963 0.82 EGFR (0.48) EGFRKDR
SCHEMBL21750828 0.82 EGFR (0.54) EGFRKDR
SCHEMBL17934393 0.81 EGFR (0.55) EGFRKDR
SCHEMBL17934408 0.81 EGFR (0.57) EGFRKDR
SCHEMBL21751018 0.81 EGFR (0.53) EGFRKDR
SCHEMBL21750943 0.81 EGFR (0.48) EGFRKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246328-B1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR, AND PREPARATION AND APPLICATION THEREOF BEIJING SCITECH MQ PHARMACEUTICALS LTD (CN) 2020-07-22 EP disclosed
EP-3246328-B1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR, AND PREPARATION AND APPLICATION THEREOF BEIJING SCITECH MQ PHARMACEUTICALS LTD (CN) 2020-07-22 EP disclosed
US-10106508-B2 Quinazoline heterocyclic compound as EGFR kinase inhibitor and preparation and application thereof BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2018-10-23 US disclosed
US-20170355683-A1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR AND PREPARATION AND APPLICATION THEREOF BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2017-12-14 US disclosed
US-20170355683-A1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR AND PREPARATION AND APPLICATION THEREOF BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2017-12-14 US disclosed
US-20170355683-A1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR AND PREPARATION AND APPLICATION THEREOF BEIJING SCITECH-MQ PHARMACEUTICALS LIMITED (CN) 2017-12-14 US disclosed
EP-3246328-A1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR, AND PREPARATION AND APPLICATION THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2017-11-22 EP disclosed
EP-3246328-A1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR, AND PREPARATION AND APPLICATION THEREOF Beijing Scitech-MQ Pharmaceuticals Limited (CN) 2017-11-22 EP disclosed
WO-2016112847-A1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR, AND PREPARATION AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2016-07-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170355683-A1 QUINAZOLINE HETEROCYCLIC COMPOUND AS EGFR KINASE INHIBITOR AND PREPARATION AND APPLICATION THEREOF EGFR, ERBB2, ERBB4 EGFR 1/4885KDR 85/4885
US-10106508-B2 Quinazoline heterocyclic compound as EGFR kinase inhibitor and preparation and application thereof EGFR, ERBB2, ERBB4 EGFR 1/4885KDR 85/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.