SCHEMBL1797133

SCHEMBL1797133

Cc1cc(-c2cncc(F)c2)cc(C(=O)Nc2cccc(C#N)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 1/20 0.49
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
ATR Q13535 1/20 0.46
ALDH1A1 P00352 2/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
SCN10A Q9Y5Y9 3/20 0.45
SCN2A Q99250 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C9 P11712 2/20 0.45
GRM5 P41594 1/20 0.45
KCNH2 Q12809 1/20 0.44
CYP3A4 P08684 1/20 0.44
POLB P06746 1/20 0.44
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1794822 0.91 GRM4 (0.54) GRM4NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL1792836 0.86 ATR (0.59) GRM4NPC1RAB9ASMN1; SMN2ATR
SCHEMBL1795347 0.85 CYP1A2 (0.48) GRM4NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL1792907 0.85 CYP1A2 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1SCN10A
SCHEMBL1798210 0.82 HSD17B10 (0.51) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL1795787 0.82 SMN1; SMN2 (0.52) NPC1RAB9ASMN1; SMN2ALDH1A1SCN10A
SCHEMBL1798303 0.81 GRM4 (0.62) GRM4NPC1RAB9ASMN1; SMN2ATR
SCHEMBL1793853 0.80 CYP1A2 (0.50) CYP1A2CYP2C9GRM5CYP3A4
SCHEMBL1798156 0.78 CYP1A2 (0.48) CYP1A2CYP2C9GRM5KCNH2CYP3A4
SCHEMBL1794776 0.78 LRRK2 (0.47) GRM4SCN10ASCN2AGRM5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed