SCHEMBL17976152

SCHEMBL17976152

C[C@H](NC(=O)c1ccc2c(c1)/C(=C(/Nc1ccc(CN3CCCCC3)cc1)c1ccccc1)C(=O)N2)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
RAB9A P51151 1/20 0.47
GRK5 P34947 9/20 0.45
MCHR1 Q99705 6/20 0.43
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
PAK4 O96013 2/20 0.42
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17976080 1.00 GAA (0.47) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976082 1.00 GAA (0.47) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976154 1.00 GAA (0.47) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976455 0.95 GRK5 (0.43) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976307 0.95 GRK5 (0.47) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976454 0.95 GRK5 (0.43) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976205 0.95 GRK5 (0.43) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976208 0.95 GRK5 (0.43) GAAHTTRAB9AGRK5MCHR1
SCHEMBL17976310 0.95 GRK5 (0.47) GAAHTTRAB9AGRK5MCHR1
SCHEMBL6974280 0.94 HTT (0.48) GAAHTTRAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO claimed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP claimed
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO disclosed
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO disclosed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP disclosed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP disclosed