SCHEMBL17976469

SCHEMBL17976469

CCN(CC)Cc1ccc(N/C(=C2\C(=O)Nc3ccc(C(=O)OC)cc32)c2ccncc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
AKT2 P31751 1/20 0.40
PDPK1 O15530 2/20 0.39
NAMPT P43490 3/20 0.39
PDGFRB P09619 1/20 0.39
KIT P10721 1/20 0.39
KDR P35968 1/20 0.39
ROCK2 O75116 2/20 0.38
AURKA O14965 1/20 0.38
RAF1 P04049 1/20 0.38
CHEK1 O14757 1/20 0.38
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
HDAC3 O15379 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3942421 0.93 KDM4E (0.41) KDM4EALDH1A1MAPTNAMPTCHEK1
SCHEMBL3942424 0.93 KDM4E (0.41) KDM4EALDH1A1MAPTNAMPTCHEK1
SCHEMBL17976401 0.91 AKT2 (0.41) AKT2PDPK1NAMPTROCK2CHEK1
SCHEMBL23252178 0.91 KDM4E (0.49) KDM4EALDH1A1MAPTPDPK1PDGFRB
SCHEMBL17976398 0.91 AKT2 (0.41) AKT2PDPK1NAMPTROCK2CHEK1
SCHEMBL17976127 0.90 PDPK1 (0.42) KDM4EALDH1A1MAPTAKT2PDPK1
SCHEMBL2570748 0.84 KDM4E (0.49) KDM4EALDH1A1MAPT
SCHEMBL3942241 0.84 BACE1 (0.42) KDM4EALDH1A1MAPTAKT2NAMPT
SCHEMBL3942237 0.84 BACE1 (0.42) KDM4EALDH1A1MAPTAKT2NAMPT
SCHEMBL2570750 0.84 KDM4E (0.49) KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO disclosed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP disclosed