SCHEMBL17976751

SCHEMBL17976751

CCCC(Oc1cc(C)c(-n2ccc(C(F)(F)F)n2)c(C)c1)c1ccc(C(=O)NCCC(=O)O)cc1

nearest known ligand 0.80

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GCG P01275 12/20 0.80
GCGR P47871 10/20 0.76
GLP1R P43220 2/20 0.76
CHRM5 P08912 1/20 0.76
GIPR P48546 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11962749 0.89 GCG (1.00) GCGGCGRGLP1RCHRM5GIPR
SCHEMBL11962691 0.87 GCGR (0.76) GCGGCGRGLP1RGIPR
SCHEMBL11962739 0.87 GCG (1.00) GCGGCGRGLP1RCHRM5
Pf-06291874 SCHEMBL11901097 0.86 GCGR (1.00) GCGGCGRGLP1RCHRM5GIPR
Pf-06291874 SCHEMBL11899337 0.86 GCGR (1.00) GCGGCGRGLP1RCHRM5GIPR
Pf-06291874 SCHEMBL11900272 0.86 GCGR (1.00) GCGGCGRGLP1RCHRM5GIPR
SCHEMBL11899682 0.81 GCG (1.00) GCGGCGRGLP1RCHRM5
SCHEMBL11899686 0.81 GCG (1.00) GCGGCGRGLP1RCHRM5
SCHEMBL16310832 0.81 GCGR (0.80) GCGGCGRGLP1RCHRM5
SCHEMBL11899926 0.81 GCG (1.00) GCGGCGRGLP1RCHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2673260-B1 GLUCAGON RECEPTOR MODULATOR PFIZER (US) 2016-08-17 EP disclosed