SCHEMBL17979324

SCHEMBL17979324

CCCc1nn(C)c2c(=O)[nH]c(-c3cc(CC4CCC4)ccc3OCC)nc12

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 18/20 0.75
HDAC6 Q9UBN7 12/20 0.75
HDAC1 Q13547 10/20 0.75
PDE3A Q14432 4/20 0.75
HDAC2 Q92769 6/20 0.67
HDAC3 O15379 3/20 0.67
NCOR2 Q9Y618 3/20 0.67
PDE6C P51160 3/20 0.66
KMT2A Q03164 2/20 0.66
PDE1A P54750 2/20 0.66
PDE1B Q01064 2/20 0.66
PDE1C Q14123 2/20 0.66
MEN1 O00255 1/20 0.66
ALDH1A1 P00352 1/20 0.66
HPGD P15428 1/20 0.66
KDM4E B2RXH2 1/20 0.63
PDE3B Q13370 2/20 0.62
PDE2A O00408 1/20 0.62
ABCC4 O15439 1/20 0.62
ABCC5 O15440 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17390153 0.93 PDE5A (0.73) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL17980848 0.90 PDE5A (0.76) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL18714950 0.90 PDE5A (0.74) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL16003753 0.88 PDE5A (0.89) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL16003676 0.88 PDE5A (0.89) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL16003761 0.88 PDE5A (0.89) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL16003783 0.88 PDE5A (0.89) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL17390102 0.88 PDE5A (0.84) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL18715295 0.88 PDE5A (0.70) PDE5AHDAC6HDAC1PDE3AHDAC2
SCHEMBL16003653 0.88 PDE5A (0.77) PDE5AHDAC6HDAC1PDE3AHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016120432-A1 COMPOUNDS AND METHODS FOR ANTICOAGULATION THERAPY FUNDACIÓN PARA LA INVESTIGACIÓN MÉDICA APLICADA (ES) 2016-08-04 WO disclosed