SCHEMBL17980850

SCHEMBL17980850

CCCc1nn(C)c2c(=O)[nH]c(-c3cc(C(O)c4ccc(C(N)=O)cc4)ccc3OCC)nc12

nearest known ligand 0.83

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 18/20 0.83
HDAC6 Q9UBN7 11/20 0.83
HDAC1 Q13547 11/20 0.83
HDAC2 Q92769 7/20 0.83
PDE6C P51160 2/20 0.72
KMT2A Q03164 2/20 0.64
HDAC3 O15379 1/20 0.64
NCOR2 Q9Y618 1/20 0.64
MEN1 O00255 1/20 0.62
ALDH1A1 P00352 1/20 0.62
HPGD P15428 1/20 0.62
PDE1A P54750 1/20 0.62
PDE1B Q01064 1/20 0.62
PDE1C Q14123 1/20 0.62
PDE3B Q13370 1/20 0.60
PDE3A Q14432 1/20 0.60
KDM4E B2RXH2 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17390166 0.91 PDE5A (0.84) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL16003767 0.91 PDE5A (1.00) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL17980849 0.91 PDE5A (0.83) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL18714952 0.90 PDE5A (0.85) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL18714967 0.89 PDE5A (0.82) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL25013454 0.87 PDE5A (0.74) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL18714928 0.86 PDE5A (0.84) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL18714940 0.85 PDE5A (0.83) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL30848755 0.84 PDE5A (0.71) PDE5AHDAC6HDAC1HDAC2PDE6C
SCHEMBL7961020 0.84 PDE5A (1.00) PDE5AHDAC6HDAC1HDAC2PDE6C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016120432-A1 COMPOUNDS AND METHODS FOR ANTICOAGULATION THERAPY FUNDACIÓN PARA LA INVESTIGACIÓN MÉDICA APLICADA (ES) 2016-08-04 WO disclosed