SCHEMBL18012007

SCHEMBL18012007

CNC(=O)c1cnc(Nc2ccccc2)nc1Nc1cccc(NC(=O)OC(C)(C)C)c1

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.63
EGFR P00533 11/20 0.59
BTK Q06187 6/20 0.59
MET P08581 2/20 0.55
JAK3 P52333 2/20 0.51
MAPK8 P45983 1/20 0.50
MAPK9 P45984 1/20 0.50
ALK Q9UM73 1/20 0.49
ITK Q08881 6/20 0.49
BRD4 O60885 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18011892 0.91 SYK (0.66) SYKEGFRBTKJAK3MAPK8
SCHEMBL14769149 0.87 BTK (0.64) SYKEGFRBTKMETJAK3
SCHEMBL13498136 0.86 EGFR (0.59) SYKEGFRBTKITK
SCHEMBL14769279 0.86 EGFR (0.69) SYKEGFRBTKJAK3ITK
SCHEMBL18012019 0.86 SYK (0.60) SYKEGFRBTKJAK3ITK
SCHEMBL12519750 0.85 BTK (0.77) SYKEGFRBTKJAK3ITK
SCHEMBL14679200 0.84 SYK (0.60) SYKEGFRBTKMAPK8MAPK9
SCHEMBL13074512 0.84 SYK (0.60) SYKEGFRBTKMETMAPK8
SCHEMBL13166506 0.83 SYK (0.67) SYKEGFRBTKJAK3ITK
SCHEMBL18357348 0.83 EGFR (0.59) SYKEGFRBTKJAK3MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016124160-A1 PYRIMIDOPYRIMIDINEDIONE DERIVATIVES AS EGFR INHIBITORS AND APPLICATION THEREOF 华东理工大学 2016-08-11 WO disclosed