SCHEMBL18025751

SCHEMBL18025751

COc1cccc(C2C(=O)Nc3ccccc32)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.55
PDE4B Q07343 1/20 0.55
PDE4C Q08493 1/20 0.55
PDE4D Q08499 1/20 0.55
DDB1 Q16531 1/20 0.49
CRBN Q96SW2 1/20 0.49
KDM4E B2RXH2 5/20 0.47
GAA P10253 4/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
NPC1 O15118 3/20 0.47
ALDH1A1 P00352 5/20 0.46
HPGD P15428 3/20 0.46
GLA P06280 1/20 0.46
HTR7 P34969 1/20 0.46
LMNA P02545 1/20 0.44
GPR174 Q9BXC1 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GID4 Q8IVV7 1/20 0.43
MAPT P10636 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3968527 0.85 CDYL (0.50) PDE4APDE4BPDE4CPDE4DDDB1
SCHEMBL18025745 0.84 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DDDB1
SCHEMBL16641809 0.82 PDE4A (0.44) PDE4APDE4BPDE4CPDE4D
SCHEMBL13431421 0.81 BRD4 (0.51) PDE4APDE4BPDE4CPDE4DDDB1
SCHEMBL18025771 0.81 MAPT (0.49) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6385829 0.80 DDB1 (0.55) DDB1CRBNKDM4EGAAMEN1
SCHEMBL31728057 0.78 IDO1 (0.51) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL2828597 0.78 IDO1 (0.51) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL6930683 0.78 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DKDM4E
SCHEMBL16634786 0.78 MAPT (0.49) PDE4APDE4BPDE4CPDE4DGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016133217-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE OXINDOLE COMPOUND AND TRIAZOLIUM SALT USED THEREIN AS CATALYST 国立大学法人名古屋大学 2016-08-25 WO disclosed