SCHEMBL18036554

SCHEMBL18036554

Cc1ccncc1-c1ccc(NS(C)(=O)=O)cc1C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 14/20 0.65
PTGS2 P35354 3/20 0.43
PTGS1 P23219 2/20 0.43
DHODH Q02127 1/20 0.41
NAMPT P43490 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL526764 0.88 CYP17A1 (0.69) CYP17A1PTGS2PTGS1
SCHEMBL526869 0.84 CYP17A1 (0.70) CYP17A1PTGS2PTGS1
SCHEMBL526391 0.84 CYP17A1 (0.78) CYP17A1PTGS2PTGS1
SCHEMBL15733042 0.84 CYP17A1 (0.51) CYP17A1PTGS2PTGS1DHODHNAMPT
SCHEMBL526755 0.81 CYP17A1 (0.76) CYP17A1PTGS2PTGS1
SCHEMBL10273708 0.80 CYP17A1 (0.65) CYP17A1PTGS2PTGS1
SCHEMBL526580 0.79 CYP17A1 (0.76) CYP17A1PTGS2PTGS1
SCHEMBL527331 0.79 CYP17A1 (1.00) CYP17A1
SCHEMBL16277425 0.78 DHODH (0.48) DHODH
SCHEMBL527098 0.78 CYP17A1 (1.00) CYP17A1PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598481-B1 SULFONAMIDE COMPOUNDS USEFUL AS CYP17 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2016-08-31 EP claimed