Tyrosine

Tyrosine

SCHEMBL180585

CSCCC(N)C(=O)O.NC(Cc1ccc(O)cc1)C(=O)O

nearest known ligand 0.71

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.71
PTGS1 P23219 2/20 0.51
ALPI P09923 1/20 0.51
PKM P14618 1/20 0.51
XIAP P98170 1/20 0.51
HIF1A Q16665 2/20 0.49
KDM4E B2RXH2 1/20 0.49
USP2 O75604 1/20 0.49
EGFR P00533 1/20 0.49
LCK P06239 1/20 0.49
FYN P06241 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
ALOX15 P16050 1/20 0.49
HTR2A P28223 1/20 0.49
PTGS2 P35354 1/20 0.49
RECQL P46063 1/20 0.49
HSD17B10 Q99714 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
TPH1 P17752 1/20 0.46
GRB2 P62993 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tyrosine SCHEMBL28430992 1.00 SLC7A5 (0.71) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL180587 1.00 SLC7A5 (0.71) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL27531942 0.93 SLC7A5 (0.61) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL7764501 0.93 SLC7A5 (0.65) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL7764495 0.93 SLC7A5 (0.65) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL1724134 0.92 SLC7A5 (0.60) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL27625516 0.92 SLC7A5 (0.60) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL28477318 0.91 SLC7A5 (0.58) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL8630269 0.91 SLC7A5 (0.58) SLC7A5PTGS1ALPIPKMXIAP
Tyrosine SCHEMBL1585313 0.91 SLC7A5 (0.58) SLC7A5PTGS1ALPIPKMXIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200353088-A1 PEPTIDE CONJUGATE CGRP RECEPTOR ANTAGONISTS AND METHODS OF PREPARATION AND USES THEREOF AUCKLAND UNISERVICES LIMITED (NZ) 2020-11-12 US claimed
EP-3707157-A1 PEPTIDE CONJUGATE CGRP RECEPTOR ANTAGONISTS AND METHODS OF PREPARATION AND USES THEREOF Auckland Uniservices Limited (NZ) 2020-09-16 EP claimed
CN-111479823-A Peptide conjugate CGRP receptor antagonist and preparation method and application thereof 奥克兰联合服务有限公司 2020-07-31 CN claimed
US-20200353088-A1 PEPTIDE CONJUGATE CGRP RECEPTOR ANTAGONISTS AND METHODS OF PREPARATION AND USES THEREOF AUCKLAND UNISERVICES LIMITED (NZ) 2020-11-12 US disclosed
EP-3707157-A1 PEPTIDE CONJUGATE CGRP RECEPTOR ANTAGONISTS AND METHODS OF PREPARATION AND USES THEREOF Auckland Uniservices Limited (NZ) 2020-09-16 EP disclosed
CN-111479823-A Peptide conjugate CGRP receptor antagonist and preparation method and application thereof 奥克兰联合服务有限公司 2020-07-31 CN disclosed
CN-110234346-A Novel vaccine against Zika virus and combination of DNA antibody constructs for use against Zika virus 宾夕法尼亚大学理事会 2019-09-13 CN disclosed
WO-2019078697-A2 ANTI-CD3 ANTIBODY AND PHARMACEUTICAL COMPOSITION FOR CANCER TREATMENT COMPRISING SAME 주식회사 녹십자 2019-04-25 WO disclosed
US-20150111816-A1 METHODS AND TREATMENT WITH GLP-1 RECEPTOR AGONISTS PHASEBIO PHARMACEUTICALS, INC. (US) 2015-04-23 US disclosed
US-20140364362-A1 THERAPEUTIC AGENTS COMPRISING INSULIN AMINO ACID SEQUENCES PHASEBIO PHARMACEUTICALS INC (US) 2014-12-11 US disclosed
EP-2400974-A2 SYNTHETIC DIBLOCK COPOLYPEPTIDE HYDROGELS FOR USE IN THE CENTRAL NERVOUS SYSTEM The Regents Of The University Of California (US) 2012-01-04 EP disclosed
WO-2010096572-A2 SYNTHETIC DIBLOCK COPOLYPEPTIDE HYDROGELS FOR USE IN THE CENTRAL NERVOUS SYSTEM THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-08-26 WO disclosed
EP-1750521-A1 METHOD AND SYSTEM FOR SOLUBILIZING PROTEIN The Texas A&M University System (US) 2007-02-14 EP disclosed
WO-2005117602-A1 METHOD AND SYSTEM FOR SOLUBILIZING PROTEIN THE TEXAS A & M UNIVERSITY SYSTEM (US) 2005-12-15 WO disclosed
US-5062935-A METHOD OF VAPORIZING A SAMPLE SUBSTANCE BRUKER-FRANZEN ANALYTIK GMBH (DE) 1991-11-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200353088-A1 PEPTIDE CONJUGATE CGRP RECEPTOR ANTAGONISTS AND METHODS OF PREPARATION AND USES THEREOF CALCRL, CALCR, GRPR SLC7A5 1069/4885PTGS1 1469/4885ALPI 2106/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.