SCHEMBL1806715

SCHEMBL1806715

CSc1ccc2c(c1)c(CCN)c(C)n2Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.70
CYP3A4 P08684 2/20 0.70
CYP2C19 P33261 2/20 0.70
CYP2D6 P10635 1/20 0.70
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
PNMT P11086 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
PLA2G2A P14555 7/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.38
CCR2 P41597 3/20 0.37
MEN1 O00255 1/20 0.37
RGS12 O14924 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
PKM P14618 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19064528 0.90 CYP1A2 (0.71) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL19064530 0.86 CYP1A2 (0.66) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL19064549 0.86 CYP1A2 (0.76) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL19064543 0.86 CYP1A2 (0.69) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL16027044 0.82 CYP1A2 (1.00) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL19064533 0.81 CYP1A2 (0.78) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
Hydrochloric Acid SCHEMBL19064529 0.81 CYP1A2 (0.98) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL19088169 0.77 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL19064532 0.76 CYP1A2 (0.78) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1
SCHEMBL9960009 0.76 CYP1A2 (0.53) CYP1A2CYP3A4CYP2C19CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011060976-A1 TRYPTAMINE-DERIVED COMPOUNDS AS ANTIBACTERIAL AGENTS UNIVERSITE DE LIEGE (BE) 2011-05-26 WO claimed
WO-2011060976-A1 TRYPTAMINE-DERIVED COMPOUNDS AS ANTIBACTERIAL AGENTS UNIVERSITE DE LIEGE (BE) 2011-05-26 WO disclosed