SCHEMBL1809270

SCHEMBL1809270

CN(C)Cc1ccc(S(N)(=O)=O)cc1Nc1ncnc2cc(OCCCN3CCOCC3)ccc12.CNS(=O)(=O)c1ccc(N(C)C)c(Nc2ncnc3cc([N+](=O)[O-])ccc23)c1

nearest known ligand 0.75

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRAF P15056 15/20 0.75
TNNI3K Q59H18 15/20 0.75
HRH3 Q9Y5N1 1/20 0.43
SRC P12931 1/20 0.43
KDR P35968 1/20 0.43
EGFR P00533 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1804731 0.86 BRAF (0.67) BRAFTNNI3KHRH3SRCKDR
SCHEMBL6911431 0.86 BRAF (1.00) BRAFTNNI3KSRCKDR
Hydrochloric Acid SCHEMBL1805208 0.86 BRAF (0.98) BRAFTNNI3KSRCKDR
SCHEMBL6910959 0.77 TNNI3K (0.85) BRAFTNNI3K
Hydrochloric Acid SCHEMBL12006441 0.76 TNNI3K (0.84) BRAFTNNI3K
SCHEMBL6912894 0.75 BRAF (0.77) BRAFTNNI3KSRCKDREGFR
SCHEMBL24777171 0.75 TNNI3K (0.88) BRAFTNNI3K
SCHEMBL1810590 0.74 TNNI3K (1.00) BRAFTNNI3KSRCKDREGFR
SCHEMBL1806419 0.74 BRAF (0.64) BRAFTNNI3KHRH3KDREGFR
SCHEMBL29606885 0.74 TNNI3K (0.85) BRAFTNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501233-A1 QUINAZOLINE COMPOUNDS GlaxoSmithKline LLC (US) 2012-09-26 EP claimed
WO-2011056740-A1 QUINAZOLINE COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-05-12 WO claimed
EP-2501233-A1 QUINAZOLINE COMPOUNDS GlaxoSmithKline LLC (US) 2012-09-26 EP disclosed
WO-2011056740-A1 QUINAZOLINE COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-05-12 WO disclosed