SCHEMBL18102986

SCHEMBL18102986

COc1cc(C=C2SC(=S)N(CC(=O)O)C2=O)ccc1OCC(=O)O

nearest known ligand 0.87

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 3/20 0.87
MEN1 O00255 6/20 0.79
KMT2A Q03164 6/20 0.79
POLB P06746 3/20 0.79
PTPN1 P18031 1/20 0.79
DUSP3 P51452 1/20 0.73
BLM P54132 1/20 0.73
PTPN5 P54829 1/20 0.73
PTPN11 Q06124 1/20 0.73
TDP1 Q9NUW8 1/20 0.73
ADAMTS5 Q9UNA0 1/20 0.69
PDE4B Q07343 1/20 0.69
GFER P55789 2/20 0.68
CASP6 P55212 1/20 0.68
NPC1 O15118 1/20 0.68
MAPK1 P28482 1/20 0.68
CTNNB1 P35222 2/20 0.67
TCF4 P15884 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18102842 1.00 AKR1B1 (0.87) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL10592653 0.96 AKR1B1 (0.89) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL10492241 0.93 AKR1B1 (0.85) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL10492234 0.93 AKR1B1 (0.85) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL12008446 0.90 CTNNB1 (0.77) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL19999083 0.89 MEN1 (0.75) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL18102840 0.89 AKR1B1 (0.76) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL19736251 0.88 AKR1B1 (1.00) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL29408611 0.88 AKR1B1 (1.00) AKR1B1MEN1KMT2APOLBPTPN1
SCHEMBL6720207 0.88 AKR1B1 (1.00) AKR1B1MEN1KMT2APOLBPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016154255-A1 INHIBITORS OF THE NOTCH TRANSCRIPTIONAL ACTIVATION COMPLEX AND METHODS FOR USE OF THE SAME UNIVERSITY OF MIAMI (US) 2016-09-29 WO disclosed