SCHEMBL18156435

SCHEMBL18156435

Cc1cccc2c(=O)[nH]c(-c3ccc(CN4CCC(O[SiH](c5ccccc5)C(C)(C)C)CC4)cc3)cc12

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TNKS O95271 16/20 0.63
PARP1 P09874 3/20 0.63
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
KDR P35968 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16616797 0.82 TNKS (0.63) TNKSPARP1OPRM1OPRK1KDR
SCHEMBL16616339 0.79 TNKS (0.78) TNKSPARP1
SCHEMBL15775242 0.78 TNKS (0.83) TNKSPARP1
SCHEMBL16625125 0.78 TNKS (1.00) TNKSPARP1
Hydrochloric Acid SCHEMBL15775374 0.77 TNKS (0.81) TNKSPARP1
SCHEMBL15775444 0.77 TNKS (0.81) TNKSPARP1
SCHEMBL16625120 0.76 TNKS (0.77) TNKSPARP1
SCHEMBL16625111 0.76 TNKS (1.00) TNKSPARP1
SCHEMBL16616588 0.76 TNKS (1.00) TNKSPARP1
SCHEMBL16625108 0.75 TNKS (1.00) TNKSPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2822656-B1 3-ARYL-5-SUBSTITUTED-ISOQUINOLIN-1-ONE COMPOUNDS AND THEIR THERAPEUTIC USE CANCER RES INST ROYAL (GB) 2016-10-19 EP disclosed