SCHEMBL18156472

SCHEMBL18156472

CNC(=O)c1ccc(-c2cc3c(C)cc(F)cc3c(=O)[nH]2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 7/20 0.53
RIPK1 Q13546 1/20 0.44
PARP1 P09874 6/20 0.41
PARP2 Q9UGN5 1/20 0.41
CHEK1 O14757 1/20 0.41
TNKS2 Q9H2K2 2/20 0.41
CRBN Q96SW2 1/20 0.38
HDAC3 O15379 1/20 0.37
ERBB2 P04626 1/20 0.37
KDR P35968 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16625238 0.78 TNKS (0.74) TNKSRIPK1PARP1TNKS2
SCHEMBL16625250 0.75 TNKS (0.52) TNKSPARP1
SCHEMBL16625259 0.74 TNKS (0.47) TNKSPARP1TNKS2
SCHEMBL16625248 0.74 TNKS (0.54) TNKSPARP1TNKS2
SCHEMBL16625240 0.74 TNKS (0.61) TNKSPARP1
SCHEMBL16625251 0.73 TNKS (0.57) TNKSPARP1TNKS2
SCHEMBL16625236 0.73 MCHR1 (0.47) TNKSPARP1TNKS2
SCHEMBL16625264 0.72 TNKS (0.49) TNKSPARP1PARP2TNKS2
SCHEMBL16625234 0.72 TNKS (0.52) TNKSPARP1PARP2TNKS2
SCHEMBL16625242 0.72 TNKS (0.53) TNKSPARP1TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2822656-B1 3-ARYL-5-SUBSTITUTED-ISOQUINOLIN-1-ONE COMPOUNDS AND THEIR THERAPEUTIC USE CANCER RES INST ROYAL (GB) 2016-10-19 EP disclosed