SCHEMBL18172365

SCHEMBL18172365

CC(C)(C)NC(=O)c1cc(-c2ccc(C(F)(F)F)cc2)cc(-n2nnnc2C(C)(C)C)c1.CC(C)(C)NC(=O)c1cc(-c2ccc(Cl)c(F)c2)cc(-n2nnnc2C(C)(C)C)c1.CC(C)(C)NC(=O)c1cc(-c2ccc(F)c(F)c2)cc(-n2nnnc2C(C)(C)C)c1.Cc1cc(-c2cc(C(=O)NC(C)(C)C)cc(-n3nnnc3C(C)(C)C)c2)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 13/20 0.45
LMNA P02545 2/20 0.34
OPRD1 P41143 2/20 0.33
ALOX5AP P20292 2/20 0.33
FEN1 P39748 2/20 0.33
TMEM97 Q5BJF2 1/20 0.33
KCNH2 Q12809 1/20 0.33
HSD11B1 P28845 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
SCN9A Q15858 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18172441 0.89 P2RY14 (0.40) P2RY14HSD11B1MAPTSCN9A
SCHEMBL18172398 0.88 P2RY14 (0.40) P2RY14LMNAHSD11B1MAPT
SCHEMBL18172506 0.86 P2RY14 (0.41) P2RY14ALOX5APFEN1HSD11B1MAPT
SCHEMBL18172487 0.86 P2RY14 (0.56) P2RY14LMNAOPRD1TMEM97KCNH2
SCHEMBL18172456 0.86 P2RY14 (0.41) P2RY14OPRD1TMEM97KCNH2SCN9A
SCHEMBL18172390 0.83 P2RY14 (0.35) P2RY14KCNH2SCN9A
SCHEMBL18172392 0.83 P2RY14 (0.40) P2RY14LMNATP53MAPT
SCHEMBL18172356 0.82 P2RY14 (0.35) P2RY14LMNA
SCHEMBL18172409 0.81 P2RY14 (0.42) P2RY14KCNH2HSD11B1TP53MAPT
SCHEMBL18172495 0.80 P2RY14 (0.36) P2RY14LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286182-A1 TETRAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PSYCHIATRIC DISORDERS F. Hoffmann-La Roche AG (CH) 2018-02-28 EP disclosed
WO-2016169902-A1 TETRAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PSYCHIATRIC DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2016-10-27 WO disclosed