SCHEMBL18174824

SCHEMBL18174824

[2H]C([2H])(C)N1C(=N)N[C@](C)(c2cc(NC(=O)c3ccc(OC)cn3)cc(F)c2F)CS1(=O)=O

nearest known ligand 0.56

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.56
BACE2 Q9Y5Z0 7/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18174823 0.95 BACE1 (0.51) BACE1BACE2
SCHEMBL18174821 0.92 BACE1 (0.56) BACE1BACE2
SCHEMBL18174825 0.90 BACE1 (0.57) BACE1BACE2
SCHEMBL18174826 0.90 BACE1 (0.45) BACE1BACE2
SCHEMBL10328883 0.88 BACE1 (0.59) BACE1BACE2
SCHEMBL10328897 0.88 BACE1 (0.57) BACE1BACE2
SCHEMBL18174828 0.88 BACE1 (0.44) BACE1BACE2
SCHEMBL18174822 0.87 BACE1 (0.52) BACE1BACE2
SCHEMBL18174816 0.87 BACE1 (0.51) BACE1BACE2
SCHEMBL15892967 0.86 BACE1 (0.57) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9475785-B2 Iminothiadiazine dioxide compounds as BACE inhibitors, compositions and their use MERCK SHARP & DOHME CORP. (US) 2016-10-25 US disclosed