Bromide

Bromide

SCHEMBL1817816

Br.Cc1cc(=O)oc2cc(NC(=O)[C@@H](N)CCCNC(N)=O)ccc12

nearest known ligand 0.58

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.54
CA1 P00915 3/20 0.54
CA9 Q16790 3/20 0.54
KDM4E B2RXH2 7/20 0.52
ALDH1A1 P00352 7/20 0.52
HPGD P15428 6/20 0.52
RAB9A P51151 5/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
NPC1 O15118 4/20 0.52
HSD17B10 Q99714 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 3/20 0.51
GAA P10253 2/20 0.51
GLA P06280 1/20 0.51
CASP3 P42574 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2230757 0.91 CA12 (0.53) CA12CA1CA9KDM4EALDH1A1
SCHEMBL7209462 0.91 CA12 (0.53) CA12CA1CA9KDM4EALDH1A1
SCHEMBL29543705 0.91 CA12 (0.53) CA12CA1CA9KDM4EALDH1A1
Hydrochloric Acid SCHEMBL380910 0.90 CA12 (0.52) CA12CA1CA9KDM4EALDH1A1
Hydrochloric Acid SCHEMBL5314266 0.90 CA12 (0.52) CA12CA1CA9KDM4EALDH1A1
Acetic Acid SCHEMBL5968184 0.89 CA12 (0.53) CA12CA1CA9KDM4EALDH1A1
Acetic Acid SCHEMBL30688431 0.89 CA12 (0.53) CA12CA1CA9KDM4EALDH1A1
SCHEMBL18220742 0.88 CA12 (0.60) CA12CA1CA9KDM4EALDH1A1
Hydrochloric Acid SCHEMBL29805418 0.88 CA12 (0.49) CA12CA1CA9KDM4EALDH1A1
SCHEMBL31130790 0.88 KDM4E (0.58) CA12CA1CA9KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12492422-B2 Ex vivo protease activity detection for disease detection/diagnostic, staging, monitoring and treatment Sunbird Bio, Inc. (US) 2025-12-09 US disclosed
US-20250297300-A1 DETECTION, STAGING, MONITORING AND TREATING A DISEASE OR A CONDITION Sunbird Bio, Inc. 2025-09-25 US disclosed
US-20250223627-A1 FLUOROGENIC SUBSTRATES FOR AMINOPEPTIDASE DETECTION IN BIOFLUIDS Sunbird Bio, Inc. 2025-07-10 US disclosed
US-20250215476-A1 EX VIVO PROTEASE ACTIVITY DETECTION FOR HEPATOCELLULAR CARCINOMA Sunbird Bio, Inc. 2025-07-03 US disclosed
US-20250197917-A1 METHOD OF PROTEASE DETECTION Sunbird Bio, Inc. 2025-06-19 US disclosed
US-12305217-B2 Ex vivo protease activity detection for disease detection/diagnostic, staging, monitoring and treatment Sunbird Bio, Inc. (US) 2025-05-20 US disclosed
US-20250110130-A1 EX VIVO PROTEASE ACTIVATION AND DETECTION Sunbird Bio, Inc. 2025-04-03 US disclosed
US-20250092437-A1 DISEASE DETECTION WITH COMBINATORIAL BIOMARKERS Sunbird Bio, Inc. 2025-03-20 US disclosed
US-11851697-B2 Ex vivo protease activity detection for disease detection/diagnostic, staging, monitoring and treatment GLYMPSE BIO, INC. (US) 2023-12-26 US disclosed
US-20230175037-A1 EX VIVO PROTEASE ACTIVITY DETECTION FOR DISEASE DETECTION/DIAGNOSTIC, STAGING, MONITORING AND TREATMENT Sunbird Bio, Inc. 2023-06-08 US disclosed
US-20220178935-A1 EX VIVO PROTEASE ACTIVITY DETECTION FOR DISEASE DETECTION/DIAGNOSTIC, STAGING, MONITORING AND TREATMENT Sunbird Bio, Inc. 2022-06-09 US disclosed
US-20220128567-A1 EX VIVO PROTEASE ACTIVITY DETECTION FOR DISEASE DETECTION/DIAGNOSTIC, STAGING, MONITORING AND TREATMENT Sunbird Bio, Inc. 2022-04-28 US disclosed
US-20220128546-A1 EX VIVO PROTEASE ACTIVITY DETECTION FOR DISEASE DETECTION/DIAGNOSTIC, STAGING, MONITORING AND TREATMENT Sunbird Bio, Inc. 2022-04-28 US disclosed
US-9526753-B2 Preparation comprising amino acids and plants and its activity in the alcohol detoxification MODUTECH S.A. (CH) 2016-12-27 US disclosed
US-9192638-B2 Preparation comprising amino acids and plants and its activity in the alcohol detoxification MODUTECH S.A. (CH) 2015-11-24 US disclosed
US-20140220162-A1 PREPARATION COMPRISING AMINO ACIDS AND PLANTS AND ITS ACTIVITY IN THE ALCOHOL DETOXIFICATION Hangzhou Adamerck Pharmlabs Inc. (CN) 2014-08-07 US disclosed
EP-2493488-B1 PREPARATION COMPRISING AMINO ACIDS AND PLANTS AND ITS ACTIVITY IN THE ALCOHOL DETOXIFICATION AND TREATING MIGRAINE MODUTECH S A (CH) 2014-01-15 EP disclosed
US-20120269909-A1 PREPARATION COMPRISING AMINO ACIDS AND PLANTS AND ITS ACTIVITY IN THE ALCOHOL DETOXIFICATION Hangzhou Adamerck Pharmlabs Inc. (CN) 2012-10-25 US disclosed
EP-2493488-A1 PREPARATION COMPRISING AMINO ACIDS AND PLANTS AND ITS ACTIVITY IN THE ALCOHOL DETOXIFICATION Modutech S.A. (CH) 2012-09-05 EP disclosed
WO-2011051900-A1 PREPARATION COMPRISING AMINO ACIDS AND PLANTS AND ITS ACTIVITY IN THE ALCOHOL DETOXIFICATION MODUTECH S.A. (CH) 2011-05-05 WO disclosed