SCHEMBL18183147

SCHEMBL18183147

C/C(=C\c1ccccc1)[C@H]1C[C@@H]1N[C@H]1CC[C@H](NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 13/20 0.73
MAOB P27338 1/20 0.62
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
DRD2 P14416 2/20 0.41
KCNA3 P22001 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18182597 1.00 KDM1A (0.73) KDM1AMAOBKMT2AL3MBTL1NFKB1
SCHEMBL18182985 1.00 KDM1A (0.73) KDM1AMAOBKMT2AL3MBTL1NFKB1
SCHEMBL18182141 1.00 KDM1A (0.73) KDM1AMAOBKMT2AL3MBTL1NFKB1
SCHEMBL18182633 1.00 KDM1A (0.73) KDM1AMAOBKMT2AL3MBTL1NFKB1
SCHEMBL18182674 0.87 KDM1A (0.56) KDM1AMAOBKMT2AL3MBTL1NFKB1
SCHEMBL18181821 0.86 KDM1A (0.64) KDM1AMAOBKMT2AL3MBTL1DRD2
SCHEMBL18183001 0.86 KDM1A (0.64) KDM1AMAOBKMT2AL3MBTL1DRD2
SCHEMBL18181896 0.86 KDM1A (0.64) KDM1AMAOBKMT2AL3MBTL1DRD2
SCHEMBL21088918 0.85 KDM1A (0.55) KDM1AMAOBKMT2AL3MBTL1NFKB1
SCHEMBL18173026 0.85 KDM1A (0.86) KDM1AMAOBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016172496-A1 LSD1 INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS, INC. (US) 2016-10-27 WO disclosed