SCHEMBL18192829

SCHEMBL18192829

O=C(O)NC1=NC2(c3cc(NC(=O)c4ccc(Cl)cn4)ccc3F)COCC2CS1

nearest known ligand 0.70

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.70
BACE2 Q9Y5Z0 9/20 0.70
KCNH2 Q12809 2/20 0.61
CYP2D6 P10635 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18192877 1.00 BACE1 (0.70) BACE1BACE2KCNH2CYP2D6
SCHEMBL933409 0.93 BACE1 (0.80) BACE1BACE2KCNH2CYP2D6
SCHEMBL12694642 0.93 BACE1 (0.80) BACE1BACE2KCNH2CYP2D6
SCHEMBL18192879 0.92 BACE1 (0.59) BACE1BACE2KCNH2
SCHEMBL2620122 0.89 BACE1 (0.87) BACE1BACE2KCNH2CYP2D6
SCHEMBL2932592 0.89 BACE1 (0.87) BACE1BACE2KCNH2CYP2D6
SCHEMBL18192930 0.87 BACE1 (0.66) BACE1BACE2KCNH2CYP2D6
SCHEMBL18192869 0.87 BACE1 (0.66) BACE1BACE2KCNH2CYP2D6
SCHEMBL968113 0.85 BACE1 (0.75) BACE1BACE2KCNH2CYP2D6
SCHEMBL18192909 0.85 BACE1 (0.68) BACE1BACE2KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451793-B1 BACE INHIBITORS LILLY CO ELI (US) 2016-11-02 EP disclosed