Ly-2886721

Ly-2886721

SCHEMBL18195437

NC1=N[C@@]2(c3cc(NC(=O)c4ccc(F)cn4)ccc3F)COCC2CS1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 1.00
BACE2 Q9Y5Z0 13/20 1.00
KCNH2 Q12809 4/20 0.69
CTSD P07339 1/20 0.69
CYP2D6 P10635 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ly-2886721 SCHEMBL971344 1.00 BACE1 (1.00) BACE1BACE2KCNH2CTSDCYP2D6
Ly-2886721 SCHEMBL966802 1.00 BACE1 (1.00) BACE1BACE2KCNH2CTSDCYP2D6
Ly-2886721 SCHEMBL30477100 1.00 BACE1 (1.00) BACE1BACE2KCNH2CTSDCYP2D6
Ly-2886721 SCHEMBL970474 0.99 BACE1 (0.98) BACE1BACE2KCNH2CTSDCYP2D6
Ly-2886721 SCHEMBL31235710 0.99 BACE1 (0.98) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2620122 0.93 BACE1 (0.87) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2932592 0.93 BACE1 (0.87) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL3306806 0.91 BACE1 (0.84) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2620249 0.91 BACE1 (0.84) BACE1BACE2KCNH2CTSDCYP2D6
SCHEMBL2965834 0.91 BACE1 (0.84) BACE1BACE2KCNH2CTSDCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451793-B1 BACE INHIBITORS LILLY CO ELI (US) 2016-11-02 EP disclosed