SCHEMBL18197830

SCHEMBL18197830

Nc1cc(CO)c2ccc(Br)cc2n1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.50
ACHE P22303 1/20 0.42
CHEK1 O14757 1/20 0.41
MPO P05164 1/20 0.41
PABPC1 P11940 2/20 0.40
HRH4 Q9H3N8 1/20 0.38
HTT P42858 1/20 0.37
TYMS P04818 1/20 0.36
PDPK1 O15530 1/20 0.36
JAK2 O60674 1/20 0.36
MEN1 O00255 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 1/20 0.36
F2 P00734 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13907108 0.83 BACE1 (0.50) BACE1ACHEMPOPABPC1HRH4
SCHEMBL8141994 0.79 CHEK1 (0.41) BACE1ACHECHEK1MPOHRH4
SCHEMBL20880351 0.79 BACE1 (0.44) BACE1ACHEHRH4
SCHEMBL832149 0.78 BACE1 (0.58) BACE1ACHEHTTTYMSRAB9A
SCHEMBL13906869 0.76 BACE1 (0.41) BACE1ACHEMPOHRH4HTT
SCHEMBL17646468 0.75 BACE1 (0.59) BACE1ACHEF2
SCHEMBL11346168 0.75 BACE1 (0.53) BACE1ACHEMPOPABPC1HRH4
SCHEMBL4257660 0.73 BACE1 (0.47) BACE1ACHE
SCHEMBL22233563 0.73 KMT2A (0.45) BACE1KMT2AMAPT
SCHEMBL21556304 0.73 F2 (0.39) CHEK1MPOHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3567035-A1 N-SUBSTITUTED 2,5-DIOXO-AZOLINE COMPOUNDS FOR USE IN THE TREATMENT OF CANCER Canbas Co. Ltd. (JP) 2019-11-13 EP disclosed
EP-3088397-A1 COMPOUNDS THAT ABROGATE THE CELL CYCLE G2 CHECKPOINT FOR USE IN THE TREATMENT OF CANCER Canbas Co. Ltd. (JP) 2016-11-02 EP disclosed