SCHEMBL181989

SCHEMBL181989

CN(C(=O)OC(C)(C)C)[C@H]1CCN(C(=O)N[C@@H](CCc2ccccc2)C(=O)N2CCC(N3C(=O)C(C)(C)c4ccccc43)CC2)C1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.38
TACR2 P21452 1/20 0.38
TACR1 P25103 1/20 0.38
HSD11B1 P28845 2/20 0.37
CACNA1B Q00975 6/20 0.37
CALCRL Q16602 1/20 0.37
CCKBR P32239 1/20 0.37
KMT2A Q03164 2/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3623022 0.91 TACR2 (0.44) TACR2TACR1CACNA1BCALCRLCCKBR
SCHEMBL181885 0.90 TACR2 (0.41) TACR2TACR1CACNA1BCALCRLCCKBR
SCHEMBL181884 0.90 TACR2 (0.41) TACR2TACR1CACNA1BCALCRLCCKBR
SCHEMBL181920 0.88 CALCRL (0.41) TACR2TACR1CACNA1BCALCRLCCKBR
SCHEMBL181919 0.88 CALCRL (0.41) TACR2TACR1CACNA1BCALCRLCCKBR
SCHEMBL180948 0.87 KMT2A (0.47) CALCRLCCKBRKMT2AMAPK1
SCHEMBL180947 0.87 KMT2A (0.47) CALCRLCCKBRKMT2AMAPK1
SCHEMBL181580 0.83 CALCRL (0.41) TACR2TACR1CACNA1BCALCRLCCKBR
SCHEMBL181581 0.83 CALCRL (0.41) TACR2TACR1CACNA1BCALCRLCCKBR
SCHEMBL182025 0.83 CALCRL (0.41) TACR2TACR1CACNA1BCALCRLCCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2401268-A1 OXYINDOLE DERIVATIVES WITH MOTILIN RECEPTOR AGONISTIC ACTIVITY RaQualia Pharma Inc (JP) 2012-01-04 EP disclosed