SCHEMBL18203296

SCHEMBL18203296

Nc1ncnc2c1nc(Sc1cc3c(cc1-c1ccco1)CCCS3)n2CCC1CCN(C=O)CC1

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.60
HSP90AB1 P08238 20/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11909105 0.97 HSP90AA1 (0.62) HSP90AA1HSP90AB1
SCHEMBL18203454 0.88 HSP90AA1 (0.62) HSP90AA1HSP90AB1
SCHEMBL18203516 0.87 HSP90AA1 (0.60) HSP90AA1HSP90AB1
SCHEMBL18169542 0.87 HSP90AA1 (0.64) HSP90AA1HSP90AB1
SCHEMBL18203481 0.87 HSP90AA1 (0.61) HSP90AA1HSP90AB1
SCHEMBL11908793 0.86 HSP90AA1 (0.63) HSP90AA1HSP90AB1
SCHEMBL18203291 0.83 HSP90AA1 (0.57) HSP90AA1HSP90AB1
SCHEMBL11908150 0.82 HSP90AA1 (0.77) HSP90AA1HSP90AB1
SCHEMBL1669387 0.80 HSP90AA1 (0.62) HSP90AA1HSP90AB1
SCHEMBL1670397 0.79 HSP90AA1 (0.60) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3091019-B1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2019-04-03 EP disclosed
EP-3091019-A2 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS Sloan Kettering Institute For Cancer Research (US) 2016-11-09 EP disclosed