SCHEMBL18211331

SCHEMBL18211331

Cc1cc(N[SH](=O)=O)ccc1/C=C/S(=O)(=O)N1CCC2(CC1)N=C(c1cccc(OC(F)(F)F)c1)NC2=O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 6/20 0.41
SCN9A Q15858 3/20 0.35
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
KIT P10721 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
PIM1 P11309 1/20 0.32
OTUD7B Q6GQQ9 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16087580 1.00 PTH1R (0.41) PTH1RSCN9ACCNT1CDK9HCRTR1
SCHEMBL16302254 0.93 PTH1R (0.37) PTH1R
SCHEMBL848059 0.92 PTH1R (0.43) PTH1RSCN9ACCNT1CDK9KIT
SCHEMBL848058 0.92 PTH1R (0.43) PTH1RSCN9ACCNT1CDK9KIT
SCHEMBL879962 0.91 PTH1R (0.43) PTH1RSCN9ACCNT1CDK9HCRTR1
SCHEMBL848151 0.90 PTH1R (0.42) PTH1RSCN9ACCNT1CDK9KIT
SCHEMBL848149 0.90 PTH1R (0.42) PTH1RSCN9ACCNT1CDK9KIT
SCHEMBL13555176 0.89 PTH1R (0.43) PTH1RSCN9ACCNT1CDK9MMP2
SCHEMBL847449 0.88 PTH1R (0.45) PTH1RSCN9AHCRTR1HCRTR2MMP2
SCHEMBL847448 0.88 PTH1R (0.45) PTH1RSCN9AHCRTR1HCRTR2MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9487517-B2 Spiroimidazolone derivative CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2016-11-08 US disclosed