SCHEMBL18213680

SCHEMBL18213680

Cc1ccc(C2(C(=O)Nc3ccc4[nH]c(C(C)(C)C)cc4c3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 6/20 0.58
MAPT P10636 3/20 0.45
NPSR1 Q6W5P4 2/20 0.45
HTR1E P28566 1/20 0.45
S1PR3 Q99500 1/20 0.45
LMNA P02545 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
POLB P06746 1/20 0.44
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
MAOA P21397 4/20 0.41
MAOB P27338 4/20 0.41
HDAC1 Q13547 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK14 Q16539 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23506675 0.96 CFTR (0.56) CFTRMAPTNPSR1HTR1ES1PR3
SCHEMBL19752874 0.95 CFTR (0.56) CFTRMAPTNPSR1HTR1ES1PR3
SCHEMBL12741439 0.91 CFTR (0.58) CFTRMAPTNPSR1LMNASMN1; SMN2
SCHEMBL23506855 0.90 CFTR (0.57) CFTRMAOAMAOBHDAC1THRB
SCHEMBL12741328 0.90 CFTR (0.57) CFTRMAPTNPSR1LMNAMEN1
SCHEMBL23836906 0.89 MAPT (0.56) CFTRMAPTNPSR1HTR1ES1PR3
SCHEMBL1465627 0.88 CFTR (0.75) CFTRMAPTNPSR1LMNAKMT2A
SCHEMBL19753053 0.87 CFTR (0.55) CFTRMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL12741185 0.87 CFTR (0.56) CFTRHPGDMAOAMAOBHDAC1
SCHEMBL12741655 0.87 CFTR (0.56) CFTRMAPTMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3091011-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Inc. (US) 2016-11-09 EP disclosed