SCHEMBL18235563

SCHEMBL18235563

CC(C)(C)OC(=O)N1CCCC(n2nc(-c3ccc(Oc4ccccc4)nc3)c3c(N)ncnc32)C1

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.76
BLK P51451 2/20 0.75
ITK Q08881 2/20 0.75
FGR P09769 1/20 0.75
FLT3 P36888 1/20 0.75
CSK P41240 1/20 0.75
JAK3 P52333 1/20 0.75
EGFR P00533 1/20 0.64
LCK P06239 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177356 1.00 BTK (0.76) BTKBLKITKFGRFLT3
SCHEMBL20177257 0.95 BTK (0.76) BTKBLKITKFGRFLT3
SCHEMBL20177246 0.95 BTK (0.76) BTKBLKITKFGRFLT3
SCHEMBL29671300 0.92 BTK (0.81) BTKBLKITKFGRFLT3
SCHEMBL15641034 0.92 BTK (0.81) BTKBLKITKFGRFLT3
SCHEMBL30324920 0.92 BTK (0.81) BTKBLKITKFGRFLT3
SCHEMBL1628863 0.92 BTK (0.81) BTKBLKITKFGRFLT3
SCHEMBL12808088 0.92 BTK (0.81) BTKBLKITKFGRFLT3
SCHEMBL21338869 0.91 BTK (0.76) BTKBLKITKFGRFLT3
SCHEMBL24197246 0.91 BTK (0.71) BTKBLKITKFGRFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016180334-A1 DUAL-SITE IRREVERSIBLE BRUTON'S TYROSINE KINASE INHIBITOR, COMPOSITION AND APPLICATION THEREFOF 杭州和正医药有限公司 2016-11-17 WO disclosed