SCHEMBL18235655

SCHEMBL18235655

OCc1ccc(Oc2ccc(Cl)c(C(F)(F)F)c2)c(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.52
IDO1 P14902 2/20 0.49
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
S1PR1 P21453 1/20 0.43
SCN9A Q15858 3/20 0.43
PLA2G7 Q13093 4/20 0.42
FFAR1 O14842 2/20 0.41
TTR P02766 2/20 0.40
CSF1R P07333 1/20 0.40
RET P07949 1/20 0.40
PDGFRB P09619 1/20 0.40
KIT P10721 1/20 0.40
PDGFRA P16234 1/20 0.40
DDR1 Q08345 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17884222 0.92 AR (0.52) ARIDO1PPARGPPARAS1PR1
SCHEMBL14656196 0.89 AR (0.50) ARIDO1PPARGPPARAS1PR1
SCHEMBL29918343 0.89 AR (0.50) ARIDO1PPARGPPARAS1PR1
SCHEMBL14670088 0.88 AR (0.49) ARIDO1PPARGPPARAS1PR1
SCHEMBL17884223 0.88 AR (0.52) ARIDO1PPARGPPARAS1PR1
SCHEMBL29918384 0.85 IDO1 (0.50) ARIDO1PPARGPPARAS1PR1
SCHEMBL875664 0.85 IDO1 (0.50) ARIDO1PPARGPPARAS1PR1
SCHEMBL29918437 0.85 AR (0.67) ARPLA2G7
SCHEMBL875787 0.85 AR (0.67) ARPLA2G7
SCHEMBL932893 0.83 IDO1 (0.61) IDO1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016180247-A1 BICYCLIC COMPOUND USED AS AN LP-PLA2 INHIBITOR, AND PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 中国科学院上海药物研究所 2016-11-17 WO disclosed