SCHEMBL1824352

SCHEMBL1824352

c1coc(-c2ccc3ncnc(Nc4ccc(-n5cncn5)cc4)c3c2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 7/20 0.49
DYRK1A Q13627 1/20 0.48
EGFR P00533 1/20 0.46
CYP1A2 P05177 4/20 0.46
CYP3A4 P08684 4/20 0.46
LMNA P02545 3/20 0.46
USP2 O75604 3/20 0.46
CYP2D6 P10635 3/20 0.46
TSHR P16473 3/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 2/20 0.46
CYP2C19 P33261 2/20 0.46
KMT2A Q03164 2/20 0.46
PI4KB Q9UBF8 1/20 0.46
CD38 P28907 3/20 0.46
HIF1A Q16665 2/20 0.44
MAPK1 P28482 3/20 0.43
RAF1 P04049 2/20 0.43
BRAF P15056 1/20 0.43
MAP4K4 O95819 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13292198 0.84 BRAF (0.59) CLK4EGFRCYP1A2CYP3A4LMNA
SCHEMBL4890693 0.81 PI4KB (0.68) CLK4DYRK1AEGFRCYP1A2CYP3A4
SCHEMBL1824255 0.81 EGFR (0.50) CLK4DYRK1AEGFRCYP1A2CYP3A4
SCHEMBL1824864 0.80 RIPK2 (0.60) CD38MAP4K4
SCHEMBL1823059 0.80 KDM4E (0.61) EGFRCYP1A2CYP3A4LMNACYP2D6
SCHEMBL1823364 0.79 MAPT (0.64) CLK4EGFRCYP1A2CYP3A4LMNA
SCHEMBL1823186 0.79 PIK3CA (0.61) CLK4DYRK1AEGFRCYP1A2CYP3A4
SCHEMBL1823225 0.79 MAPT (0.48) EGFRLMNAMEN1ALDH1A1KMT2A
SCHEMBL29450569 0.78 RAF1 (0.58) CLK4EGFRCYP1A2CYP3A4LMNA
SCHEMBL1825395 0.78 EGFR (0.52) CLK4EGFRCYP1A2CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981876-B1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS ARROW THERAPEUTICS LTD (GB) 2011-05-04 EP disclosed