Erythromycin Ethylsuccinate

Erythromycin Ethylsuccinate

SCHEMBL18259

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nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

rplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Erythromycin Ethylsuccinate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 10/20 1.00
SLCO1B3 Q9NPD5 3/20 1.00
SLCO1B1 Q9Y6L6 3/20 1.00
USP2 O75604 3/20 1.00
PGR P06401 1/20 0.88
HTR1A P08908 1/20 0.88
DRD1 P21728 1/20 0.88
SLC6A2 P23975 1/20 0.88
OPRM1 P35372 1/20 0.88
DRD3 P35462 1/20 0.88
SLC6A3 Q01959 1/20 0.88
KCNH2 Q12809 5/20 0.79
ABCB1 P08183 2/20 0.79
TSHR P16473 2/20 0.79
LMNA P02545 2/20 0.79
TDP1 Q9NUW8 1/20 0.79
MLNR O43193 1/20 0.79
ALB P02768 1/20 0.79
CNR1 P21554 1/20 0.79
HTR2A P28223 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Erythromycin Ethylsuccinate SCHEMBL537373 1.00 CYP3A4 (1.00) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL7866739 1.00 CYP3A4 (1.00) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL5082211 1.00 CYP3A4 (1.00) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL9807840 0.99 CYP3A4 (0.99) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL15665988 0.99 CYP3A4 (0.99) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL10673952 0.99 CYP3A4 (0.99) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL9118779 0.99 CYP3A4 (0.99) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL10382844 0.99 CYP3A4 (0.99) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL7750959 0.99 CYP3A4 (0.98) CYP3A4SLCO1B3SLCO1B1USP2PGR
Erythromycin Ethylsuccinate SCHEMBL7755531 0.98 CYP3A4 (0.97) CYP3A4SLCO1B3SLCO1B1USP2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 62166 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250228841-A1 COMPOSITIONS AFFECTING PIGMENT PRODUCTION AND METHODS FOR TREATMENT OF BACTERIAL DISEASES APTORUM THERAPEUTICS LTD (HK) 2025-07-17 US claimed
CN-114641296-B Preparation of an Ananamycin Liposome precursor lyophilized 德州大学系统董事会 2025-05-27 CN claimed
US-12285471-B2 Methods for treating pulmonary disease using inter-alpha inhibitor proteins PROTHERA BIOLOGICS, INC. (US) 2025-04-29 US claimed
CN-114444363-B Method, device and equipment for calculating response of high-precision receiver at any position 中南大学 2024-11-19 CN claimed
CN-118873548-A Anti-liver cancer cell preparation and application thereof 新乡医学院 2024-11-01 CN claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
CN-118510533-A Cancer diagnostic method using ephrin B2 expression 血管基因治疗公司 2024-08-16 CN claimed
CN-118389556-A Perforin preparation method and application thereof 复旦大学附属中山医院 2024-07-26 CN claimed
EP-3464579-B1 COMPOSITIONS COMPRISING POLYPEPTIDES HAVING GALACTANASE ACTIVITY AND POLYPEPTIDES HAVING BETA-GALACTOSIDASE ACTIVITY NOVOZYMES AS (DK) 2024-07-17 EP claimed
EP-3925601-B1 GASTRO-RESISTANT FORMULATION CONTAINING POSACONAZOLE AND A POLYMERIC PRECIPITATION INHIBITOR TIEFENBACHER ALFRED E GMBH & CO KG (DE) 2024-07-17 EP claimed
EP-0005238-A2 Floor covering for indoor or outdoor sporting and playing areas Schmidt, Bernard L. (US) 1979-11-14 EP claimed
EP-0004578-A1 Pellets containing styrene polymer and aluminium hydroxide, and process for preparing flame-retarding styrene polymer foams HOECHST AKTIENGESELLSCHAFT (DE) 1979-10-17 EP claimed
EP-0004587-A2 Polyvinyl alcohol pellets containing a plasticizer, and method for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1979-10-17 EP claimed
EP-0003752-A1 Process for preparing molecular-sieve-containing grains having good mechanical solidity, the grains manufactured by this process and their use Kali-Chemie Aktiengesellschaft (DE) 1979-09-05 EP claimed
WO-1979000606-A1 PROCESS FOR OBTAINING ALUMINIUM BY ELECTROLYSIS IN A MELTED BATH VAW VER ALUMINIUM WERKE AG (DE) 1979-08-23 WO claimed
EP-0003598-A1 Process for the production of aluminium by electrolysis of fused salts VEREINIGTE ALUMINIUM-WERKE AKTIENGESELLSCHAFT (DE) 1979-08-22 EP claimed
EP-0001766-A2 Method for improving the processing qualities of powdery polyolefins HOECHST AKTIENGESELLSCHAFT (DE) 1979-05-16 EP claimed
WO-1979000132-A1 PROCESS AND DEVICE FOR THE GRANULATION OF MOLTEN MATERIALS SVENSKT STAL AB (SE) 1979-03-22 WO claimed
EP-0000357-A1 Process for the preparation of cross-linkable ethylene polymer mouldings and their use as electrical insulating materials BASF Aktiengesellschaft (DE) 1979-01-24 EP claimed
US-4076804-A Erythromycin therapy ABBOTT LABORATORIES (US) 1978-02-28 US claimed