SCHEMBL182597

SCHEMBL182597

CNC(=O)C(OC)c1ccccc1COc1cc(C)ccc1C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.45
LMNA P02545 2/20 0.41
HTT P42858 1/20 0.41
LPAR1 Q92633 2/20 0.41
FABP4 P15090 1/20 0.41
FABP5 Q01469 1/20 0.41
ALDH1A1 P00352 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
TSHR P16473 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TDP1 Q9NUW8 2/20 0.39
GAA P10253 1/20 0.39
USP2 O75604 1/20 0.39
POLB P06746 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL230669 1.00 SMN1; SMN2 (0.45) SMN1; SMN2LMNAHTTLPAR1FABP4
SCHEMBL29371189 1.00 SMN1; SMN2 (0.45) SMN1; SMN2LMNAHTTLPAR1FABP4
SCHEMBL29365871 1.00 SMN1; SMN2 (0.45) SMN1; SMN2LMNAHTTLPAR1FABP4
SCHEMBL29368766 1.00 SMN1; SMN2 (0.45) SMN1; SMN2LMNAHTTLPAR1FABP4
SCHEMBL16858325 1.00 SMN1; SMN2 (0.45) SMN1; SMN2LMNAHTTLPAR1FABP4
SCHEMBL29354984 1.00 SMN1; SMN2 (0.45) SMN1; SMN2LMNAHTTLPAR1FABP4
Acetamide SCHEMBL28557945 0.96 MEN1 (0.42) SMN1; SMN2LMNAHTTLPAR1FABP4
SCHEMBL15402001 0.91 MRGPRX4 (0.43) SMN1; SMN2LMNALPAR1FABP4FABP5
SCHEMBL28593087 0.91 PTGDR2 (0.42) SMN1; SMN2LMNAHTTLPAR1FABP4
SCHEMBL7524475 0.89 SMN1; SMN2 (0.44) SMN1; SMN2LMNAHTTLPAR1FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2074 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118102874-A Active compound combinations and fungicide compositions comprising them 拜耳公司 2024-05-28 CN claimed
US-20230413824-A1 AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2023-12-28 US claimed
EP-4250926-A1 AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI Industries Ltd. (IN) 2023-10-04 EP claimed
CN-116801720-A Novel agrochemical compositions comprising 3-substituted benzamidine compounds and uses thereof 皮埃企业有限公司 2023-09-22 CN claimed
CN-116725007-A Oily liquid fungicidal formulations 阿达玛马克西姆股份有限公司 2023-09-12 CN claimed
US-20230276804-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING PYRAZOLOPYRIDINE ANTHRANILAMIDE COMPOUND, OXIDES OR SALTS THEREOF PI INDUSTRIES LTD. (IN) 2023-09-07 US claimed
US-20230276803-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING THIETANYLOXY COMPOUND, OXIDES OR SALTS THEREOF PI INDUSTRIES LTD. (IN) 2023-09-07 US claimed
CN-109152357-B Oily liquid fungicidal formulations 阿达玛马克西姆股份有限公司 2023-09-05 CN claimed
CN-116669554-A Use of Dhodh inhibitors for controlling resistant phytopathogenic fungi in crops 拜耳公司 2023-08-29 CN claimed
EP-4188094-A1 A PESTICIDALLY ACTIVE MIXTURE COMPRISING PYRAZOLOPYRIDINE ANTHRANILAMIDE COMPOUND, OXIDES OR SALTS THEREOF PI Industries Ltd. (IN) 2023-06-07 EP claimed
WO-2012082548-A2 SOYBEAN EVENT SYHT0H2 AND COMPOSITIONS AND METHODS FOR DETECTION THEREOF SYNGENTA PARTICIPATIONS AG (CH) 2012-06-21 WO claimed
WO-2012082542-A2 SOYBEAN EVENT SYHT04R AND COMPOSITIONS AND METHODS FOR DETECTION THEREOF SYNGENTA PARTICIPATIONS AG (CH) 2012-06-21 WO claimed
US-20120046323-A1 Use of Succinate Dehydrogenase Inhibitors and/or Respiratory Chain Complex III Inhibitors for Improving the Ratio of Harmful to Beneficial Microorganisms BAYER CROPSCIENCE AG (DE) 2012-02-23 US claimed
WO-2012013590-A2 USE OF SUCCINATE DEHYDROGENASE INHIBITORS AND/OR RESPIRATORY CHAIN COMPLEX III INHIBITORS FOR IMPROVING THE RATIO OF HARMFUL TO BENEFICIAL MICROORGANISMS BAYER CROPSCIENCE AG (DE) 2012-02-02 WO claimed
WO-2012004221-A2 ANTHRANILAMIDES IN COMBINATION WITH FUNGICIDES BAYER CROPSCIENCE AG (DE) 2012-01-12 WO claimed
US-20120010073-A1 Anthranilamides in combination with fungicides BAYER CROPSCIENCE AG (DE) 2012-01-12 US claimed
US-20110124501-A1 Active compound combinations BAYER CROPSCIENCE AG (DE) 2011-05-26 US claimed
WO-2011029506-A1 3-[1-(3-HALOALKYL)-TRIAZOLYL]-PHENYL-SULFIDE DERIVATIVES FOR USE AS ACARICIDES AND INSECTICIDES BAYER CROPSCIENCE AG (DE) 2011-03-17 WO claimed
WO-2011020567-A1 3-TRIAZOLYLPHENYL-SUBSTITUTED SULFIDE DERIVATIVES FOR USE AS ACARICIDES AND INSECTICIDES BAYER CROPSCIENCE AG (DE) 2011-02-24 WO claimed
EP-1183948-A1 STROBILURIN FUNGICIDE COMPOSITION REDUCED IN CHEMICAL DAMAGE SHIONOGI & CO., LTD. (JP) 2002-03-06 EP claimed