SCHEMBL18263245

SCHEMBL18263245

[CH]1CCCC2(C1)CCCNC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 8/20 0.39
CYP3A4 P08684 8/20 0.39
ALDH1A1 P00352 7/20 0.39
CYP1A2 P05177 5/20 0.39
USP2 O75604 4/20 0.39
HSD17B10 Q99714 5/20 0.38
TSHR P16473 2/20 0.38
CYP2C9 P11712 2/20 0.36
MAPK1 P28482 4/20 0.35
CYP2C19 P33261 3/20 0.35
HPGD P15428 2/20 0.35
TP53 P04637 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CHEK1 O14757 1/20 0.32
AURKA O14965 1/20 0.32
RPS6KA5 O75582 1/20 0.32
CHEK2 O96017 1/20 0.32
ABL1 P00519 1/20 0.32
LCK P06239 1/20 0.32
FYN P06241 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17107677 0.91 CYP2D6 (0.39) CYP2D6CYP3A4ALDH1A1CYP1A2USP2
SCHEMBL14810515 0.79 CYP2D6 (0.34) CYP2D6CYP3A4ALDH1A1CYP1A2USP2
SCHEMBL20719299 0.79 CYP2D6 (0.40) CYP2D6CYP3A4ALDH1A1CYP1A2USP2
SCHEMBL1627317 0.79
SCHEMBL165883 0.77 CYP2D6 (0.42) CYP2D6CYP3A4ALDH1A1CYP1A2USP2
SCHEMBL1793924 0.75 CYP2D6 (0.41) CYP2D6CYP3A4ALDH1A1CYP1A2USP2
SCHEMBL1796659 0.75
SCHEMBL1545685 0.75
Water SCHEMBL6402454 0.75 CYP3A4 (0.41) CYP2D6CYP3A4ALDH1A1CYP1A2USP2
SCHEMBL5428129 0.75 CYP2D6 (0.41) CYP2D6CYP3A4ALDH1A1CYP1A2USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016190847-A1 SUBSTITUTED HETEROARYL COMPOUNDS AND METHODS OF USE CALITOR SCIENCES, LLC (US) 2016-12-01 WO disclosed