SCHEMBL18266366

SCHEMBL18266366

Cc1cc(C(C)NC(=O)c2ccnc(NC(=O)C3CC3)n2)ccc1OC[C@@H](C)F

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.40
KCNB1 Q14721 2/20 0.40
ACACB O00763 5/20 0.38
PDE2A O00408 4/20 0.38
CYP3A4 P08684 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
JAK1 P23458 1/20 0.35
ABL1 P00519 1/20 0.35
TYK2 P29597 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2716024 0.95 ACACB (0.43) IDH1KCNB1ACACBPDE2A
SCHEMBL18266671 0.90 ACACB (0.38) IDH1KCNB1ACACBPDE2AJAK1
SCHEMBL2718552 0.88 ACACB (0.43) KCNB1ACACB
SCHEMBL2715541 0.85 ACACB (0.43) IDH1KCNB1ACACBPDE2ACYP3A4
SCHEMBL2717025 0.84 ACACB (0.40) IDH1KCNB1ACACBPDE2A
SCHEMBL18266576 0.84 GSK3B (0.48) ACACB
SCHEMBL18266686 0.84 ACACB (0.41) ACACBABL1
SCHEMBL2718587 0.84 ACACB (0.43) ACACBJAK1ABL1
SCHEMBL18266756 0.83 ABL1 (0.43) IDH1ACACBPDE2AJAK1ABL1
SCHEMBL2713163 0.82 ACACB (0.41) ACACBABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed