SCHEMBL18266830

SCHEMBL18266830

Cc1cc(OCC(C)F)ccc1C(C)NC(=O)c1ccnc(NC(=O)C2CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.48
MAPT P10636 10/20 0.48
GSK3A P49840 8/20 0.47
ABL1 P00519 1/20 0.46
ACACB O00763 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2715129 0.95 GSK3B (0.48) GSK3BMAPTGSK3AABL1ACACB
SCHEMBL2714930 0.85 GSK3B (0.47) GSK3BMAPTGSK3AABL1ACACB
SCHEMBL18266756 0.84 ABL1 (0.43) ABL1ACACB
SCHEMBL18266845 0.84 GSK3B (0.49) GSK3BMAPTGSK3A
SCHEMBL2715936 0.84 GSK3B (0.44) GSK3BMAPTGSK3AACACB
SCHEMBL2716280 0.83 MAPT (0.56) GSK3BMAPTACACB
SCHEMBL18266576 0.82 GSK3B (0.48) GSK3BMAPTGSK3AACACB
SCHEMBL18266823 0.81 GSK3B (0.48) GSK3BMAPTGSK3AACACB
SCHEMBL2717273 0.79 GSK3B (0.54) GSK3BMAPTGSK3A
SCHEMBL2714481 0.79 ABL1 (0.43) ABL1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed