SCHEMBL1827678

SCHEMBL1827678

COc1ccc(-n2ccc(C(=O)O)c2-c2ccc(C(N)=O)cc2C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.43
CA2 P00918 3/20 0.43
PARP10 Q53GL7 2/20 0.43
PARP1 P09874 2/20 0.43
PARP2 Q9UGN5 1/20 0.43
PARP4 Q9UKK3 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.40
MAPKAPK2 P49137 3/20 0.39
MAPT P10636 1/20 0.39
MAP4K4 O95819 1/20 0.38
PLAU P00749 1/20 0.38
PLAT P00750 1/20 0.38
KDM4E B2RXH2 2/20 0.37
PTPN11 Q06124 2/20 0.37
POLB P06746 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
CHEK2 O96017 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1950261 0.87 PTPN11 (0.42) CA1CA2PARP10PARP1PARP2
SCHEMBL242923 0.86 PTPN11 (0.46) CA1CA2PARP10PARP1PARP2
SCHEMBL1830075 0.85 SMN1; SMN2 (0.43) SMN1; SMN2MAPTKDM4EPOLBMEN1
SCHEMBL245309 0.83 SMN1; SMN2 (0.41) SMN1; SMN2MAPKAPK2PLAUPLATCHEK2
SCHEMBL249222 0.83 SMN1; SMN2 (0.41) CA1CA2PARP10PARP1PARP2
SCHEMBL242932 0.82 SMN1; SMN2 (0.41) CA1CA2PARP10PARP1PARP2
SCHEMBL244774 0.82 SMN1; SMN2 (0.41) CA1CA2PARP10PARP1PARP2
SCHEMBL243931 0.82 POLB (0.40) CA1CA2PARP10PARP1PARP2
SCHEMBL12540744 0.80 MAPT (0.45) SMN1; SMN2MAPKAPK2MAPTPLAUPLAT
SCHEMBL243838 0.79 MAPKAPK2 (0.45) MAPKAPK2MAP4K4PLAUPLATPTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2315590-A1 PYRROLE INHIBITORS OF S-NITROSOGLUTATHIONE REDUCTASE N30 Pharmaceuticals, LLC (US) 2011-05-04 EP disclosed
WO-2010019909-A1 PYRROLE INHIBITORS OF S-NITROSOGLUTATHIONE REDUCTASE N30 PHARMACEUTICALS, LLC (US) 2010-02-18 WO disclosed