SCHEMBL1829638

SCHEMBL1829638

COc1ccc2nc(C(=O)N3CCC4(CC3)CC(=O)c3cc(-c5cccnc5)ccc3O4)cc(OC)c2c1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACACB O00763 7/20 0.53
ACACA Q13085 3/20 0.48
EPHX2 P34913 1/20 0.43
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42
CYP19A1 P11511 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1827670 0.89 ACACB (0.46) ACACBACACA
SCHEMBL1830111 0.88 ACACB (0.54) ACACBACACA
SCHEMBL1829668 0.87 ACACB (0.46) ACACBACACA
SCHEMBL1830435 0.87 ACACB (0.47) ACACBACACACYP19A1
SCHEMBL1813377 0.87 ACACB (0.54) ACACBACACA
SCHEMBL1830195 0.85 ACACB (0.45) ACACBACACACYP19A1
SCHEMBL1828716 0.85 HDAC3 (0.49) ACACBACACACYP19A1
SCHEMBL1832752 0.85 ACACB (0.50) ACACBACACACYP19A1
SCHEMBL1829262 0.84 CA1 (0.44) ACACBACACACYP19A1
SCHEMBL1828229 0.84 CYP19A1 (0.46) ACACBACACACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-B1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK SHARP & DOHME (US) 2011-05-11 EP claimed