SCHEMBL18315919

SCHEMBL18315919

Cc1cc(CC(NC(=O)ON2CCC(N3Cc4ccccc4NC3=O)CC2)C(=O)N2CCC(N3CCCCC3)CC2)cc2cn[nH]c12

nearest known ligand 0.84

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 18/20 0.84
CYP3A4 P08684 10/20 0.84
CYP2D6 P10635 1/20 0.69
CALCA P06881 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18315888 0.96 CALCRL (0.78) CALCRLCYP3A4CYP2D6
SCHEMBL18315892 0.95 CALCRL (0.77) CALCRLCYP3A4CYP2D6
SCHEMBL18315945 0.93 CYP3A4 (0.85) CALCRLCYP3A4CYP2D6
SCHEMBL18315904 0.93 CALCRL (0.72) CALCRLCYP3A4CYP2D6
SCHEMBL18315889 0.93 CALCRL (0.84) CALCRLCYP3A4CYP2D6
SCHEMBL18315903 0.92 CALCRL (0.72) CALCRLCYP3A4
SCHEMBL13053544 0.92 CALCRL (1.00) CALCRLCYP3A4CYP2D6CALCA
SCHEMBL3607829 0.92 CALCRL (1.00) CALCRLCYP3A4CYP2D6CALCA
SCHEMBL18315901 0.89 CALCRL (0.84) CALCRLCYP3A4
SCHEMBL18315922 0.89 CALCRL (0.84) CALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539766-B1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2016-12-21 EP claimed