SCHEMBL18319233

SCHEMBL18319233

CC(=O)N1CCC(Oc2ccc(-c3cnc4ccccc4c3)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.52
IKBKB O14920 2/20 0.49
CHUK O15111 1/20 0.49
PIK3CD O00329 2/20 0.48
PIK3CA P42336 2/20 0.48
PIK3CB P42338 1/20 0.48
PIK3CG P48736 1/20 0.48
CYP11B2 P19099 2/20 0.47
FASN P49327 2/20 0.47
CYP4F2 P78329 1/20 0.47
CYP4A11 Q02928 1/20 0.47
MAP4K4 O95819 1/20 0.46
CSNK1G2 P78368 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
MAP4K5 Q9Y4K4 1/20 0.46
HPGDS O60760 1/20 0.45
PRMT5 O14744 1/20 0.44
NAMPT P43490 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30497889 1.00 CHEK2 (0.52) CHEK2IKBKBCHUKPIK3CDPIK3CA
Hydrochloric Acid SCHEMBL28563914 0.99 CHEK2 (0.51) CHEK2IKBKBCHUKPIK3CDPIK3CA
SCHEMBL18318598 0.89 FASN (0.52) PIK3CDPIK3CAFASNNAMPT
SCHEMBL18318292 0.89 PIK3CA (0.46) CHEK2PIK3CDPIK3CAFASNMAP4K4
SCHEMBL18318656 0.89 PIK3CA (0.56) PIK3CDPIK3CAPIK3CBPIK3CGFASN
SCHEMBL18318983 0.89 FASN (0.47) CHEK2PIK3CDPIK3CAFASNNAMPT
SCHEMBL18318670 0.89 PIK3CA (0.51) PIK3CDPIK3CAFASNNAMPT
SCHEMBL18319268 0.88 FASN (0.46) PIK3CDPIK3CAFASNMAP4K4
Hydrochloric Acid SCHEMBL18318805 0.88 FASN (0.51) PIK3CDPIK3CAFASNNAMPT
Hydrochloric Acid SCHEMBL28554846 0.88 PIK3CA (0.50) PIK3CDPIK3CAFASNNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11702388-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2023-07-18 US claimed
US-20210230116-A1 1,4-Substituted Piperidine Derivatives CEPHALON LLC 2021-07-29 US claimed
CN-107847765-B 1, 4-substituted piperidine derivatives 89生物有限公司 2021-05-04 CN claimed
EP-3310441-B1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES 89BIO LTD (IL) 2020-07-29 EP claimed
US-9902696-B2 1,4-substituted piperidine derivatives CEPHALON, INC. (US) 2018-02-27 US claimed
US-20250257035-A1 1,4-Substituted Piperidine Derivatives CEPHALON LLC 2025-08-14 US disclosed
US-12098130-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2024-09-24 US disclosed
US-20230391723-A1 1,4-Substituted Piperidine Derivatives CEPHALON LLC 2023-12-07 US disclosed
US-11702388-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2023-07-18 US disclosed
US-11702388-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2023-07-18 US disclosed
US-11702388-B2 1,4-substituted piperidine derivatives 89BIO LTD (IL) 2023-07-18 US disclosed
US-20210230116-A1 1,4-Substituted Piperidine Derivatives CEPHALON LLC 2021-07-29 US disclosed
US-20180179159-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON LLC 2018-06-28 US disclosed
US-20180179159-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON LLC 2018-06-28 US disclosed
US-9902696-B2 1,4-substituted piperidine derivatives CEPHALON, INC. (US) 2018-02-27 US disclosed
US-9902696-B2 1,4-substituted piperidine derivatives CEPHALON, INC. (US) 2018-02-27 US disclosed
US-9902696-B2 1,4-substituted piperidine derivatives CEPHALON, INC. (US) 2018-02-27 US disclosed
US-20160368874-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON LLC 2016-12-22 US disclosed
US-20160368874-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON LLC 2016-12-22 US disclosed
WO-2016205633-A1 1, 4-SUBSTITUTED PIPERIDINE DERIVATIVES CEPHALON, INC. (US) 2016-12-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250257035-A1 1,4-Substituted Piperidine Derivatives FASN, CES1, CPT1A CHEK2 4678/4885IKBKB 1701/4885CHUK 794/4885
US-20230391723-A1 1,4-Substituted Piperidine Derivatives FASN, CES1, CPT1A CHEK2 4678/4885IKBKB 1701/4885CHUK 794/4885
US-20160368874-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES FASN, CES1, CPT1A CHEK2 4678/4885IKBKB 1701/4885CHUK 794/4885
US-20210230116-A1 1,4-Substituted Piperidine Derivatives FASN, CES1, CPT1A CHEK2 4678/4885IKBKB 1701/4885CHUK 794/4885
US-11702388-B2 1,4-substituted piperidine derivatives FASN, CES1, CPT1A CHEK2 4678/4885IKBKB 1701/4885CHUK 794/4885
US-12098130-B2 1,4-substituted piperidine derivatives FASN, CES1, CPT1A CHEK2 4678/4885IKBKB 1701/4885CHUK 794/4885
US-20180179159-A1 1,4-SUBSTITUTED PIPERIDINE DERIVATIVES FASN, CES1, CPT1A CHEK2 4673/4885IKBKB 1545/4885CHUK 734/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.